SCHEMBL3383649

SCHEMBL3383649

CN(C)c1ccc(-c2ccn3c(-c4ccc(NC(=O)Nc5cccc(C(F)(F)F)c5)cc4)cnc3c2)cn1

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDR P35968 18/20 0.55
FGFR3 P22607 15/20 0.55
BRAF P15056 1/20 0.49
MAPK14 Q16539 1/20 0.49
TNNI3K Q59H18 1/20 0.49
TEK Q02763 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3186936 0.88 FGFR3 (0.56) KDRFGFR3TEK
SCHEMBL3383389 0.86 NPC1 (0.64) KDRFGFR3
SCHEMBL3386228 0.86 KDR (0.55) KDRFGFR3
SCHEMBL3190830 0.85 KDR (0.66) KDRFGFR3BRAFMAPK14TNNI3K
SCHEMBL3386132 0.84 KDR (0.55) KDRFGFR3
SCHEMBL3189323 0.82 KDR (0.59) KDRFGFR3TEK
SCHEMBL3198958 0.82 KDR (0.70) KDRFGFR3MAPK14
SCHEMBL3417464 0.81 FGFR3 (0.51) KDRFGFR3
SCHEMBL3386444 0.80 FGFR3 (0.52) KDRFGFR3
SCHEMBL13336720 0.80 KDR (0.71) KDRFGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904494-B1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS VEGF-R2 INHIBITORS LILLY CO ELI (US) 2010-12-01 EP disclosed
CN-101128461-A Imidazo (1, 2-a) pyridine compounds as VEGF-R2 inhibitors LILLY CO ELI (US) 2008-02-20 CN disclosed