SCHEMBL3384671

SCHEMBL3384671

CCOC(=O)C(C(=O)O)c1ncnc2c1ccn2S(=O)(=O)c1ccc(C)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.41
KMT2A Q03164 4/20 0.37
KDM4E B2RXH2 2/20 0.37
TSHR P16473 2/20 0.37
LMNA P02545 2/20 0.37
ALDH1A1 P00352 2/20 0.36
SLC1A3 P43003 1/20 0.36
SLC1A2 P43004 1/20 0.36
SLC1A1 P43005 1/20 0.36
RAPGEF4 Q8WZA2 1/20 0.36
PTPN11 Q06124 1/20 0.36
MEN1 O00255 2/20 0.36
POLB P06746 2/20 0.36
TP53 P04637 1/20 0.36
HPGD P15428 1/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
PIK3C3 Q8NEB9 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24262374 0.95 L3MBTL1 (0.43) L3MBTL1KMT2AKDM4ETSHRLMNA
SCHEMBL29080525 0.90 L3MBTL1 (0.46) L3MBTL1TSHRSLC1A3SLC1A2SLC1A1
SCHEMBL3384664 0.87 L3MBTL1 (0.44) L3MBTL1KMT2AKDM4EALDH1A1RAPGEF4
SCHEMBL13769391 0.80 L3MBTL1 (0.46) L3MBTL1KMT2AKDM4ETSHRLMNA
SCHEMBL30575111 0.78 L3MBTL1 (0.43) L3MBTL1KMT2AKDM4ETSHRLMNA
SCHEMBL24262373 0.78 L3MBTL1 (0.43) L3MBTL1KMT2AKDM4ETSHRLMNA
SCHEMBL4067920 0.78 L3MBTL1 (0.44) L3MBTL1KMT2AKDM4ETSHRLMNA
SCHEMBL3556162 0.76 L3MBTL1 (0.49) L3MBTL1TSHRRAPGEF4PTPN11POLB
SCHEMBL29247903 0.75 PTGDR2 (0.47) L3MBTL1KDM4ERAPGEF4PTPN11POLB
SCHEMBL13494114 0.74 L3MBTL1 (0.50) L3MBTL1TSHRALDH1A1RAPGEF4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8183248-B2 Substituted pyrrolo[2,3-d]pyrimidines and compositions as protein kinase inhibitors IRM LLC (BM) 2012-05-22 US disclosed
EP-1891066-B1 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2010-12-22 EP disclosed
US-20090118273-A1 Compounds and Compositions as Protein Kinase Inhibitors IRM LLC (BM) 2009-05-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090118273-A1 Compounds and Compositions as Protein Kinase Inhibitors SRC, FYN, SYK L3MBTL1 4367/4885KMT2A 1463/4885KDM4E 1741/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.