SCHEMBL3384948

SCHEMBL3384948

Cc1cc(F)c(C2(C)CN(C)C(=O)C(=O)N2)cc1Br

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.35
CES1 P23141 1/20 0.35
ABCC9 O60706 1/20 0.32
ABCC8 Q09428 1/20 0.32
KCNJ11 Q14654 1/20 0.32
KCNJ8 Q15842 1/20 0.32
POLB P06746 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL251389 0.90 ABCC9 (0.36) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL252703 0.81 MEN1 (0.37) ABCC9ABCC8KCNJ11KCNJ8L3MBTL1
SCHEMBL2153420 0.68 BACE1 (0.41) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL251767 0.67 ALDH1A1 (0.40)
SCHEMBL12525453 0.64 BACE1 (0.34) L3MBTL1
SCHEMBL12524922 0.62 BACE1 (0.34) L3MBTL1
SCHEMBL251000 0.61 BACE1 (0.50) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL247369 0.61 BACE1 (0.36) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9959296 0.60 BACE1 (0.38)
SCHEMBL16311227 0.60 BACE1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012000933-A1 3-AMINO-5,6-DIHYDRO-1H-PYRAZIN-2-ONE DERIVATIVES USEFUL FOR THE TREATEMENT OF ALZHEIMER'S DISEASE AND OTHER FORMS OF DEMENTIA JANSSEN PHARMACEUTICA NV (BE) 2012-01-05 WO disclosed