SCHEMBL3385282

SCHEMBL3385282

CC(C)(C)c1cc(NC(=O)NCc2ccc(-c3cnc4cc(-c5ccc(S(C)(=O)=O)cc5)ccn34)cc2F)no1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDR P35968 10/20 0.45
NTRK1 P04629 2/20 0.45
RET P07949 2/20 0.45
KCNH2 Q12809 2/20 0.45
CSF1R P07333 1/20 0.45
CCDC6 Q16204 1/20 0.45
FLT3 P36888 7/20 0.44
FGFR3 P22607 8/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3383112 0.91 RET (0.53) KDRNTRK1RETKCNH2CSF1R
SCHEMBL3383912 0.90 KDR (0.51) KDRFGFR3
SCHEMBL3385275 0.89 KDR (0.51) KDRNTRK1RETKCNH2CSF1R
SCHEMBL3383303 0.88 NPC1 (0.52) KDRNTRK1RETKCNH2CSF1R
SCHEMBL3383492 0.84 FLT3 (0.50) KDRNTRK1RETKCNH2CSF1R
SCHEMBL3383110 0.81 RET (0.48) KDRNTRK1RETKCNH2CSF1R
SCHEMBL3386505 0.81 RET (0.65) KDRNTRK1RETKCNH2CSF1R
SCHEMBL3381104 0.79 KDR (0.55) KDRNTRK1RETKCNH2CSF1R
SCHEMBL3385534 0.78 KDR (0.50) KDRRETFLT3FGFR3
SCHEMBL3381118 0.78 NPC1 (0.54) KDRRETFLT3FGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904494-B1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS VEGF-R2 INHIBITORS LILLY CO ELI (US) 2010-12-01 EP disclosed