SCHEMBL3382504

SCHEMBL3382504

CC(C)(C)c1ccnc(NC(=O)Cc2ccc(-c3cnc4cc(-c5ccncc5)ccn34)cc2F)c1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDR P35968 15/20 0.47
FGFR3 P22607 14/20 0.47
NTRK1 P04629 1/20 0.38
WNT3A P56704 1/20 0.38
FLT3 P36888 1/20 0.38
PIK3CA P42336 1/20 0.38
MTOR P42345 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3386163 0.93 WNT3A (0.42) KDRFGFR3WNT3A
SCHEMBL3383499 0.93 KDR (0.46) KDRFGFR3WNT3AFLT3PIK3CA
SCHEMBL3385818 0.93 KDR (0.49) KDRFGFR3
SCHEMBL3385477 0.91 FGFR3 (0.41) KDRFGFR3
SCHEMBL3384812 0.90 KDR (0.45) KDRFGFR3WNT3AFLT3PIK3CA
SCHEMBL3189267 0.90 KDR (0.45) KDRFGFR3WNT3A
SCHEMBL3381930 0.89 KDR (0.39) KDRFGFR3
SCHEMBL3383240 0.88 FGFR3 (0.49) KDRFGFR3WNT3A
SCHEMBL3381852 0.88 KDR (0.56) KDRFGFR3
SCHEMBL3385600 0.88 KDR (0.46) KDRFGFR3NTRK1WNT3AFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904494-B1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS VEGF-R2 INHIBITORS LILLY CO ELI (US) 2010-12-01 EP disclosed