SCHEMBL3386153

SCHEMBL3386153

CC(C)N1CCN(C(=O)c2ccc3[nH]ccc3c2)CC1.CCN1CCC(n2ccc3cc(C(=O)N4CCN(C(C)C)CC4)ccc32)C1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.45
MAPK14 Q16539 1/20 0.45
DRD2 P14416 2/20 0.43
DRD3 P35462 2/20 0.43
CCR3 P51677 1/20 0.42
HRH3 Q9Y5N1 5/20 0.42
OXTR P30559 1/20 0.41
ACHE P22303 1/20 0.40
HTR4 Q13639 1/20 0.40
LMNA P02545 1/20 0.39
GPR183 P32249 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3386037 0.91 HRH3 (0.47) HRH3
SCHEMBL3390885 0.91 HRH3 (0.47) HRH3
SCHEMBL3390881 0.90 MAPK14 (0.59) CHRM2MAPK14DRD2DRD3CCR3
SCHEMBL3390449 0.85 MAPK14 (0.57) CHRM2MAPK14DRD2DRD3CCR3
SCHEMBL3387184 0.83 HRH3 (0.44) HRH3
SCHEMBL3387192 0.83 HRH3 (0.44) HRH3
SCHEMBL3390314 0.83 HRH3 (0.44) HRH3
SCHEMBL3388360 0.83 HRH3 (0.43) CHRM2MAPK14DRD2DRD3CCR3
SCHEMBL3385812 0.81 HRH3 (0.48) HRH3OXTR
SCHEMBL3383875 0.81 DRD2 (0.52) DRD2HRH3OXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029534-B1 1H-INDOL-5-YL-PIPERAZIN-1-YL-METHANONE DERIVATIVES HOFFMANN LA ROCHE (CH) 2010-12-22 EP disclosed