SCHEMBL3386997

SCHEMBL3386997

CCCn1cc(C)c2c(=O)[nH]c(-c3ccc(OCC)c(S(=O)(=O)NCCCN4CCOCC4)c3)nc21

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 3/20 0.49
TSHR P16473 4/20 0.49
TDP1 Q9NUW8 1/20 0.49
ALDH1A1 P00352 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
HPGD P15428 1/20 0.42
BRD4 O60885 1/20 0.40
BRD2 P25440 1/20 0.40
BRD3 Q15059 1/20 0.40
KMT2A Q03164 1/20 0.40
CA12 O43570 1/20 0.40
CA9 Q16790 1/20 0.40
POLB P06746 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3017892 0.87 PDE5A (0.65) PDE5ACA12CA9POLBCYP3A4
SCHEMBL6010417 0.86 ALDH1A1 (0.48) PDE5ATSHRALDH1A1BRD4BRD2
SCHEMBL3383025 0.85 PDE5A (0.36) PDE5APOLB
SCHEMBL3029660 0.83 PDE5A (0.64) PDE5ATSHRALDH1A1L3MBTL1CA12
Hydrochloric Acid SCHEMBL3386364 0.79 PDE5A (0.48) PDE5A
SCHEMBL3023331 0.76 PDE5A (0.62) PDE5ACA12CA9
SCHEMBL3028372 0.75 PDE5A (0.63) PDE5ACA12CA9
SCHEMBL3023423 0.75 PDE5A (0.63) PDE5ACA12CA9
SCHEMBL3027989 0.74 PDE5A (0.53) PDE5A
SCHEMBL3384950 0.74 PDE5A (0.41) PDE5AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1634883-B1 2-SUBSTITUTED PHENYL-5,7-DIALKYL-3,7-DIHYDROPYRROLE[2,3-D] PYRIMIDINE-4-ONE DERIVATIVES, THE PREPARATION AND THE PHARMACEUTICAL USE THEREOF YANGTZE RIVER PHARMACEUTICAL G (CN) 2010-12-15 EP claimed
EP-1634883-A1 2-SUBSTITUTED PHENYL-5,7-DIALKYL-3,7-DIHYDROPYRROLE[2,3-D]PYRIMIDINE-4-ONE DERIVATIVES, THE PREPARATION AND THE PHARMACEUTICAL USE THEREOF Tianjin Tasly Group Co., Ltd. (CN) 2006-03-15 EP claimed