SCHEMBL3387358

SCHEMBL3387358

N#CC1(Cc2ccc(F)cc2)CCN(C(=O)C2CN(C(=O)O)c3cc(Cl)c(N)cc3O2)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
RAB9A P51151 1/20 0.33
FPR2 P25090 1/20 0.32
PROKR1 Q8TCW9 1/20 0.32
MEN1 O00255 1/20 0.30
LMNA P02545 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
HTR1A P08908 1/20 0.30
ADRA2A P08913 1/20 0.30
ADORA3 P0DMS8 1/20 0.30
CYP2C9 P11712 1/20 0.30
ADRA2B P18089 1/20 0.30
HTR2C P28335 1/20 0.30
SLC6A4 P31645 1/20 0.30
CYP2C19 P33261 1/20 0.30
DRD3 P35462 1/20 0.30
HTR2B P41595 1/20 0.30
KMT2A Q03164 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3381860 0.91 ALDH1A1 (0.37) ALDH1A1RAB9AFPR2PROKR1POLB
SCHEMBL3358997 0.89 MC4R (0.36) ALDH1A1SIRT1
SCHEMBL3352172 0.87 ALDH1A1 (0.35) ALDH1A1RAB9AFPR2PROKR1LMNA
SCHEMBL3386987 0.84 ALDH1A1 (0.34) ALDH1A1FPR2PROKR1
SCHEMBL2799068 0.84 MC4R (0.37) ALDH1A1SIRT1
SCHEMBL3355555 0.83 CCR1 (0.34) ALDH1A1RAB9AFPR2PROKR1LMNA
SCHEMBL3354707 0.83 ALDH1A1 (0.34) ALDH1A1RAB9AFPR2PROKR1POLB
SCHEMBL13330973 0.82 ALDH1A1 (0.36) ALDH1A1FPR2PROKR1MEN1LMNA
SCHEMBL3354423 0.82 LMNA (0.37) ALDH1A1FPR2PROKR1LMNA
SCHEMBL3352265 0.81 ALDH1A1 (0.33) ALDH1A1RAB9AFPR2PROKR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010068881-A1 NOVEL BENZODIOXANE AND BENZOXAZINE DERIVATIVES USEFUL AS CC CHEMOKINE RECEPTOR LIGANDS FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-06-17 WO disclosed