SCHEMBL3388862

SCHEMBL3388862

CCOc1ncnc2[nH]cnc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.40
PDPK1 O15530 2/20 0.37
TTBK1 Q5TCY1 1/20 0.34
TTBK2 Q6IQ55 1/20 0.34
CDK2 P24941 3/20 0.33
MAPK1 P28482 2/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
SLC9A1 P19634 1/20 0.33
HSD17B10 Q99714 2/20 0.33
CDC7 O00311 2/20 0.33
CDK1 P06493 2/20 0.33
TSHR P16473 2/20 0.33
PLK4 O00444 1/20 0.33
CHEK1 O14757 1/20 0.33
CHUK O15111 1/20 0.33
DYRK3 O43781 1/20 0.33
ROCK2 O75116 1/20 0.33
PRKD3 O94806 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22639807 0.84 CDK1 (0.48) KDM4EPDPK1CDK2MAPK1POLB
6-(Decyloxy)Purine SCHEMBL6234481 0.82 CDK1 (0.49) KDM4EPDPK1CDK2MAPK1POLB
SCHEMBL5175458 0.82 CDK1 (0.49) KDM4EPDPK1CDK2MAPK1POLB
SCHEMBL8937059 0.82 CDK1 (0.49) KDM4EPDPK1CDK2MAPK1POLB
SCHEMBL7027155 0.82 CDK1 (0.49) KDM4EPDPK1CDK2MAPK1POLB
SCHEMBL284829 0.81 PDPK1 (0.52) PDPK1TTBK1TTBK2MAPTLCK
SCHEMBL12270784 0.81 MAP3K7 (0.50) CDK2CDK1MAP3K7TAB1CCNB1
SCHEMBL2623129 0.80 CDK1 (0.50) CDK2CDK1MAP3K7TAB1CCNB1
SCHEMBL20322774 0.80 HSD17B10 (0.45) KDM4EHSD17B10TSHRTP53GAA
SCHEMBL31570032 0.80 PDPK1 (0.33) PDPK1CDK2MAPK1CDC7CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 109 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3131914-B1 3'-SUBSTITUTED METHYL OR ALKYNYL NUCLEOSIDES FOR THE TREATMENT OF HCV IDENIX PHARMACEUTICALS LLC (US) 2023-05-10 EP claimed
US-10202411-B2 3′-substituted methyl or alkynyl nucleosides nucleotides for the treatment of HCV IDENIX PHARMACEUTICALS LLC (US) 2019-02-12 US claimed
US-20180162898-A1 4'-OR NUCLEOSIDES FOR THE TREATMENT OF HCV IDENIX PHARMACEUTICALS LLC (US) 2018-06-14 US claimed
EP-3131914-A1 3'-SUBSTITUTED METHYL OR ALKYNYL NUCLEOSIDES FOR THE TREATMENT OF HCV Idenix Pharmaceuticals LLC (US) 2017-02-22 EP claimed
US-20170044205-A1 3'-SUBSTITUTED METHYL OR ALKYNYL NUCLEOSIDES NUCLEOTIDES FOR THE TREATMENT OF HCV IDENIX PHARMACEUTICALS, INC. 2017-02-16 US claimed
EP-3083654-A1 4'-OR NUCLEOSIDES FOR THE TREATMENT OF HCV Idenix Pharmaceuticals LLC (US) 2016-10-26 EP claimed
US-20160280729-A1 CYCLOPENTANE AND CYCLOPENTENE NUCLEOSIDE ANALOGS FOR THE TREATMENT OF HCV IDENIX PHARMACEUTICALS LLC (US) 2016-09-29 US claimed
WO-2015161137-A1 3'-SUBSTITUTED METHYL OR ALKYNYL NUCLEOSIDES FOR THE TREATMENT OF HCV IDENIX PHARMACEUTICALS, INC. (US) 2015-10-22 WO claimed
WO-2015095419-A1 4'-OR NUCLEOSIDES FOR THE TREATMENT OF HCV IDENIX PHARMACEUTICALS, INC. (US) 2015-06-25 WO claimed
WO-2015077360-A2 CYCLOPENTANE AND CYCLOPENTENE NUCLEOSIDE ANALOGS FOR THE TREATMENT OF HCV IDENIX PHARMACEUTICALS, INC. (US) 2015-05-28 WO claimed
US-20040166575-A1 Inosine producing bacterium belonging to the genus Bacillus and method for producing inosine AJINOMOTO CO., INC. (JP) 2004-08-26 US claimed
EP-1447442-A1 Inosine production by means of Bacillus bacteria able to grow in the presence of 6-ethoxypurine Ajinomoto Co., Inc. (JP) 2004-08-18 EP claimed
US-12054768-B2 Methods for detecting agglutination and compositions for use in practicing the same THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-08-06 US disclosed
EP-3131914-B1 3'-SUBSTITUTED METHYL OR ALKYNYL NUCLEOSIDES FOR THE TREATMENT OF HCV IDENIX PHARMACEUTICALS LLC (US) 2023-05-10 EP disclosed
EP-4123031-A1 METHODS FOR DETECTING AGGLUTINATION AND COMPOSITIONS FOR USE IN PRACTICING THE SAME The Regents of The University of California (US) 2023-01-25 EP disclosed
EP-3283638-B1 METHODS FOR DETECTING AGGLUTINATION AND USE OF KITS IN PRACTICING THE SAME UNIV CALIFORNIA (US) 2022-06-08 EP disclosed
EP-0421819-A1 Therapeutic nucleosides THE WELLCOME FOUNDATION LIMITED (GB) 1991-04-10 EP disclosed
EP-0417999-A1 Antiviral compounds THE WELLCOME FOUNDATION LIMITED (GB) 1991-03-20 EP disclosed
EP-0294114-A2 Antiviral compounds THE WELLCOME FOUNDATION LIMITED (GB) 1988-12-07 EP disclosed
EP-0286425-A2 Therapeutic nucleosides THE WELLCOME FOUNDATION LIMITED (GB) 1988-10-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160280729-A1 CYCLOPENTANE AND CYCLOPENTENE NUCLEOSIDE ANALOGS FOR THE TREATMENT OF HCV ZC3HAV1, HAVCR2, NSUN2 KDM4E 2632/4885PDPK1 4249/4885TTBK1 1188/4885
US-20170044205-A1 3'-SUBSTITUTED METHYL OR ALKYNYL NUCLEOSIDES NUCLEOTIDES FOR THE TREATMENT OF HCV RB1, NSUN2, METTL3 KDM4E 754/4885PDPK1 3368/4885TTBK1 2005/4885
US-10202411-B2 3′-substituted methyl or alkynyl nucleosides nucleotides for the treatment of HCV RB1, NSUN2, METTL3 KDM4E 786/4885PDPK1 3297/4885TTBK1 2003/4885
US-20180162898-A1 4'-OR NUCLEOSIDES FOR THE TREATMENT OF HCV NSUN2, NSUN3, ZC3HAV1 KDM4E 692/4885PDPK1 1891/4885TTBK1 4181/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.