SCHEMBL3388929

SCHEMBL3388929

Cc1ccc(-n2nc(C(C)(C)C)cc2N(OS(C)(=O)=O)C(=O)Nc2cnc(N3CCN(C(=O)C4(C)CC4)CC3)cc2C)cc1

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CDK8 P49336 2/20 0.34
MAPK14 Q16539 6/20 0.33
NTRK1 P04629 1/20 0.32
NTRK3 Q16288 1/20 0.32
NTRK2 Q16620 1/20 0.32
HTT P42858 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
BRAF P15056 1/20 0.32
MAPK13 O15264 3/20 0.32
MAPK12 P53778 2/20 0.32
MAPK11 Q15759 2/20 0.32
DDR2 Q16832 1/20 0.32
TNF P01375 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3390651 0.90 SMO (0.37) CDK8MAPK14HTTSMN1; SMN2KDM4E
SCHEMBL3388899 0.89 CDK8 (0.34) CDK8MAPK14BRAFMAPK13MAPK12
SCHEMBL3390498 0.87 RAB9A (0.36) CDK8MAPK14ALDH1A1BRAFMAPK13
SCHEMBL3390273 0.87 MAPK14 (0.34) CDK8MAPK14NTRK1NTRK3NTRK2
SCHEMBL3390581 0.84 P2RY12 (0.37) MAPK14SMN1; SMN2ALDH1A1
SCHEMBL3392905 0.83 SMO (0.39) CDK8MAPK14HTTSMN1; SMN2KDM4E
SCHEMBL3388924 0.82 MAPK14 (0.49) CDK8MAPK14MAPK13MAPK12MAPK11
SCHEMBL3393238 0.81 MAPK14 (0.52) CDK8MAPK14MAPK13MAPK12MAPK11
SCHEMBL3180430 0.78 CDK8 (0.35) CDK8MAPK14BRAFMAPK13MAPK12
SCHEMBL3390558 0.78 MAPK13 (0.40) MAPK14SMN1; SMN2KDM4EALDH1A1BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1943243-B1 KINASE INHIBITORS LILLY CO ELI (US) 2010-12-29 EP disclosed