SCHEMBL3392905

SCHEMBL3392905

Cc1ccc(-n2nc(C(C)(C)C)cc2N(OS(C)(=O)=O)C(=O)Nc2cnc(N3CCN(C(=O)C(C)(C)C)CC3)cc2Cl)cc1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMO Q99835 3/20 0.39
ALK Q9UM73 1/20 0.35
MAPK14 Q16539 5/20 0.35
CDK8 P49336 2/20 0.35
IKBKB O14920 1/20 0.33
PTK2 Q05397 1/20 0.33
P2RY12 Q9H244 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
DCTPP1 Q9H773 1/20 0.33
BRAF P15056 1/20 0.33
MAPK13 O15264 3/20 0.33
MAPK12 P53778 2/20 0.33
MAPK11 Q15759 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3390651 0.93 SMO (0.37) SMOMAPK14CDK8PTK2KDM4E
SCHEMBL3180430 0.87 CDK8 (0.35) MAPK14CDK8PTK2BRAFMAPK13
SCHEMBL4602880 0.85 MAPK14 (0.43) MAPK14CDK8PTK2ALDH1A1MAPK13
SCHEMBL3388929 0.83 CDK8 (0.34) MAPK14CDK8KDM4EALDH1A1GAA
SCHEMBL3392902 0.82 MAPK14 (0.52) MAPK14CDK8PTK2MAPK13MAPK12
SCHEMBL3391079 0.81 RBP4 (0.35) MAPK14CDK8PTK2P2RY12MAPK13
SCHEMBL3389956 0.80 RAB9A (0.36) MAPK14CDK8PTK2P2RY12KDM4E
SCHEMBL3392557 0.80 MAPK14 (0.54) MAPK14CDK8PTK2MAPK13MAPK12
SCHEMBL3393213 0.80 PTK2B (0.38) MAPK14PTK2KDM4ESMN1; SMN2MAPK13
SCHEMBL3393224 0.79 GBA1 (0.38) MAPK14KDM4EALDH1A1GAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1943243-B1 KINASE INHIBITORS LILLY CO ELI (US) 2010-12-29 EP disclosed