SCHEMBL3391018

SCHEMBL3391018

CC(C(=O)CC#N)(C(F)(F)F)C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 4/20 0.38
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
RIPK1 Q13546 1/20 0.31
PDK1 Q15118 1/20 0.30
PDK2 Q15119 1/20 0.30
PDK3 Q15120 1/20 0.30
PDK4 Q16654 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1011084 0.83
SCHEMBL1013569 0.82 MCL1 (0.38) MCL1CYP1A2CYP3A4CYP2C19PDK1
SCHEMBL1012319 0.81
SCHEMBL24410357 0.77 MCL1 (0.38) MCL1CYP1A2CYP3A4CYP2C19
SCHEMBL23982819 0.77 MCL1 (0.38) MCL1CYP1A2CYP3A4CYP2C19
SCHEMBL1014847 0.76 MCL1 (0.40) MCL1CYP1A2CYP3A4CYP2C19
SCHEMBL133731 0.75
SCHEMBL573401 0.75
SCHEMBL5463212 0.73 MCL1 (0.42) MCL1CYP1A2CYP2C19
SCHEMBL1583542 0.73 MCL1 (0.40) MCL1CYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1943243-B1 KINASE INHIBITORS LILLY CO ELI (US) 2010-12-29 EP disclosed