SCHEMBL3392016

SCHEMBL3392016

Fc1cccc(-c2nc3c(c(C(F)(F)F)n2)CCNC3)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 5/20 0.44
HTR2B P41595 4/20 0.44
HTR2A P28223 3/20 0.44
HTR7 P34969 2/20 0.43
ALPL P05186 1/20 0.37
ALPI P09923 1/20 0.37
GUSB P08236 1/20 0.36
ASIC3 Q9UHC3 1/20 0.36
NT5E P21589 2/20 0.36
NISCH Q9Y2I1 1/20 0.35
CYP11B2 P19099 1/20 0.34
PARP1 P09874 1/20 0.33
TNKS2 Q9H2K2 1/20 0.33
PARP2 Q9UGN5 1/20 0.33
IDO1 P14902 1/20 0.33
KDM4E B2RXH2 1/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1260880 0.99 HTR2C (0.43) HTR2CHTR2BHTR2AHTR7ALPL
SCHEMBL1967019 0.86 HTR2C (0.51) HTR2CHTR2BHTR2ASMN1; SMN2
SCHEMBL3388287 0.85 HTR2C (0.53) HTR2CHTR2BHTR2AHTR7
Hydrochloric Acid SCHEMBL1262177 0.85 HTR2C (0.50) HTR2CHTR2BHTR2ASMN1; SMN2
Hydrochloric Acid SCHEMBL1262699 0.84 HTR2A (0.52) HTR2CHTR2BHTR2AHTR7
Hydrochloric Acid SCHEMBL1262185 0.83 HTR2C (0.39) HTR2CHTR2BHTR2AHTR7ASIC3
SCHEMBL3394336 0.81 USP1 (0.43) HTR2CHTR2BHTR2APARP1KDM4E
SCHEMBL3419388 0.80 PSD (0.42) HTR2CHTR2BHTR2A
Hydrochloric Acid SCHEMBL1262796 0.80 USP1 (0.42) HTR2CHTR2BHTR2APARP1KDM4E
Hydrochloric Acid SCHEMBL1261370 0.79 PSD (0.41) HTR2CHTR2BHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863812-B1 DIPEPTIDYL PEPTIDASE-IV INHIBITING COMPOUNDS, METHODS OF PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AS AN ACTIVE AGENT LG LIFE SCIENCES LTD (KR) 2010-07-14 EP disclosed