SCHEMBL3393076

SCHEMBL3393076

COc1c[c]c(Br)c(OC)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
ALDH1A1 P00352 6/20 0.36
CYP1A2 P05177 5/20 0.36
CYP3A4 P08684 4/20 0.36
CYP1A1 P04798 4/20 0.36
CYP1B1 Q16678 4/20 0.36
POLB P06746 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CYP2E1 P05181 1/20 0.33
CYP2C8 P10632 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2A6 P11509 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP4B1 P13584 1/20 0.33
CYP2B6 P20813 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28851924 0.80 ERN1 (0.36) CA2ALDH1A1CYP3A4POLBL3MBTL1
SCHEMBL27695180 0.78 TRPV4 (0.36) ALDH1A1CYP3A4POLBL3MBTL1MAPT
SCHEMBL1810937 0.76 CA12 (0.43) CA12CA1CA2CA7CA9
SCHEMBL743497 0.76 CA12 (0.43) CA12CA1CA2CA7CA9
SCHEMBL2235124 0.74 CA12 (0.41) CA12CA1CA2CA7CA9
SCHEMBL2164088 0.74 CA12 (0.41) CA12CA1CA2CA7CA9
SCHEMBL2164186 0.74 CA12 (0.41) CA12CA1CA2CA7CA9
SCHEMBL27755946 0.74 CA12 (0.41) CA12CA1CA2CA7CA9
SCHEMBL8860398 0.71 CA12 (0.39) CA12CA1CA2CA7CA9
SCHEMBL29178171 0.71 CA1 (0.39) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112209841-B Synthesis method of terbutaline and application of terbutaline in preparation of terbutaline sulfate 扬州中宝药业股份有限公司 2022-03-04 CN claimed
CN-112209841-A Synthesis method of terbutaline and application of terbutaline in preparation of terbutaline sulfate 扬州中宝药业股份有限公司 2021-01-12 CN claimed
CN-101402623-A 3-substituted benzene phthalein compounds with biological activity SHANGHAI INST ORGANIC CHEM (CN) 2009-04-08 CN claimed
EP-3636636-B1 PYRIDONE COMPOUND AND AGRICULTURAL AND HORTICULTURAL FUNGICIDE MITSUI CHEMICALS AGRO INC (JP) 2022-07-06 EP disclosed
CN-112209841-B Synthesis method of terbutaline and application of terbutaline in preparation of terbutaline sulfate 扬州中宝药业股份有限公司 2022-03-04 CN disclosed
CN-112209841-B Synthesis method of terbutaline and application of terbutaline in preparation of terbutaline sulfate 扬州中宝药业股份有限公司 2022-03-04 CN disclosed
US-11117863-B2 Pyridone compounds and agricultural and horticultural fungicides containing the same as active ingredients MITSUI CHEMICALS AGRO, INC. (JP) 2021-09-14 US disclosed
CN-112209841-A Synthesis method of terbutaline and application of terbutaline in preparation of terbutaline sulfate 扬州中宝药业股份有限公司 2021-01-12 CN disclosed
CN-112209841-A Synthesis method of terbutaline and application of terbutaline in preparation of terbutaline sulfate 扬州中宝药业股份有限公司 2021-01-12 CN disclosed
CN-107635981-B Compounds and methods for inducing browning of white adipose tissue 中国科学院广州生物医药与健康研究院 2020-08-04 CN disclosed
US-20200172486-A1 PYRIDONE COMPOUNDS AND AGRICULTURAL AND HORTICULTURAL FUNGICIDES CONTAINING THE SAME AS ACTIVE INGREDIENTS MITSUI CHEMICALS AGRO, INC. (JP) 2020-06-04 US disclosed
EP-3636636-A1 PYRIDONE COMPOUND AND AGRICULTURAL AND HORTICULTURAL FUNGICIDE Mitsui Chemicals Agro, Inc. (JP) 2020-04-15 EP disclosed
CN-103189383-B Biaryl diphosphine ligand, its intermediate and the purposes in asymmetry catalysis thereof KANATA CHEMICAL TECHNOLOGIES INC. (CA) 2016-11-30 CN disclosed
CN-103189383-A Biaryl diphosphine ligands, intermediates of the same and their use in asymmetric catalysis KANATA CHEMICAL TECHNOLOGIES INC 2013-07-03 CN disclosed
EP-2145888-A1 Deazapurine derivatives as HSP90-Inhibitors Conforma Therapeutics Corporation (US) 2010-01-20 EP disclosed
CN-101402623-A 3-substituted benzene phthalein compounds with biological activity SHANGHAI INST ORGANIC CHEM (CN) 2009-04-08 CN disclosed
US-20070185064-A1 2-Aminopurine Analogs Having HSP90-Inhibiting Activity CONFORMA THERAPEUTICS CORPORATION (US) 2007-08-09 US disclosed
US-7138401-B2 2-aminopurine analogs having HSP90-inhibiting activity CONFORMA THERAPEUTICS CORPORATION (US) 2006-11-21 US disclosed
US-20050113340-A1 2-Aminopurine analogs having HSP90-inhibiting activity CONFORMA THERAPEUTICS CORPORATION 2005-05-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200172486-A1 PYRIDONE COMPOUNDS AND AGRICULTURAL AND HORTICULTURAL FUNGICIDES CONTAINING THE SAME AS ACTIVE INGREDIENTS PNPO, CBR3, CBR1 CA12 4431/4885CA1 2325/4885CA2 986/4885
US-20050113340-A1 2-Aminopurine analogs having HSP90-inhibiting activity HSP90AB2P, HSP90AB1, HSP90AA1 CA12 4540/4885CA1 4219/4885CA2 4096/4885
US-11117863-B2 Pyridone compounds and agricultural and horticultural fungicides containing the same as active ingredients PNPO, CBR3, CBR1 CA12 4431/4885CA1 2325/4885CA2 986/4885
US-20070185064-A1 2-Aminopurine Analogs Having HSP90-Inhibiting Activity HSP90AB2P, HSP90AB1, HSP90AA1 CA12 4540/4885CA1 4219/4885CA2 4096/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.