SCHEMBL3394397

SCHEMBL3394397

O=CC(Br)c1ccc2[nH]c3nc(Cl)ccc3c2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
GMNN O75496 1/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
PKM P14618 1/20 0.36
TSHR P16473 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
CYP2C19 P33261 1/20 0.36
MTOR P42345 1/20 0.36
BLM P54132 1/20 0.36
PMP22 Q01453 1/20 0.36
HIF1A Q16665 1/20 0.36
HSD17B10 Q99714 1/20 0.36
SIRT2 Q8IXJ6 1/20 0.35
CA5A P35218 1/20 0.33
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3395158 0.84 KDM4E (0.37) KDM4EADORA2AADORA1MAPTMEN1
SCHEMBL675608 0.76 KIF11 (0.51) KDM4EGMNNLMNACYP1A2PKM
SCHEMBL675640 0.74 PIM3 (0.45) KDM4EGMNNLMNACYP1A2PKM
SCHEMBL16241834 0.72 KDM4E (0.35) KDM4EGMNNLMNACYP1A2PKM
SCHEMBL676197 0.70 KIF11 (0.48) KDM4EGMNNLMNACYP1A2PKM
SCHEMBL676048 0.68 GSK3B (0.41) KDM4EGMNNLMNACYP1A2PKM
SCHEMBL675919 0.68 KDM4E (0.54) KDM4EGMNNLMNACYP1A2PKM
SCHEMBL676823 0.68 KDM4E (0.44) KDM4EGMNNLMNACYP1A2PKM
SCHEMBL679240 0.68 KDM4E (0.44) KDM4EGMNNLMNACYP1A2PKM
SCHEMBL675082 0.67 CA5A (0.68) KDM4EGMNNLMNACYP1A2PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010025872-A2 ALFA-CARBOLINE INHIBITORS OF NPM-ALK, RET, AND BCR-ABL UNIVERSITA' DEGLI STUDI DI MILANO-BICOCCA (IT) 2010-03-11 WO claimed
WO-2010025872-A2 ALFA-CARBOLINE INHIBITORS OF NPM-ALK, RET, AND BCR-ABL UNIVERSITA' DEGLI STUDI DI MILANO-BICOCCA (IT) 2010-03-11 WO disclosed