SCHEMBL3394947

SCHEMBL3394947

C#CCNCc1ccc(OC(F)(F)F)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PYCR1 P32322 1/20 0.54
SCN8A Q9UQD0 1/20 0.50
EPHX2 P34913 2/20 0.46
NR1H4 Q96RI1 1/20 0.46
KDM1A O60341 1/20 0.43
HTR2C P28335 3/20 0.42
ALDH1A1 P00352 2/20 0.42
TSHR P16473 1/20 0.42
PLA2G1B P04054 1/20 0.40
MAPT P10636 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ATG4B Q9Y4P1 1/20 0.40
VNN1 O95497 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8348550 0.84 SCN8A (0.55) SCN8AEPHX2NR1H4KDM1AHTR2C
Hydrochloric Acid SCHEMBL6122751 0.82 SCN8A (0.54) SCN8AEPHX2NR1H4KDM1AHTR2C
SCHEMBL3962793 0.81 SCN8A (0.54) SCN8AEPHX2NR1H4KDM1AHTR2C
SCHEMBL13527792 0.80 PYCR1 (0.79) PYCR1
SCHEMBL22729788 0.79 PYCR1 (0.61) PYCR1ALDH1A1SMN1; SMN2RAB9A
Hydrochloric Acid SCHEMBL3168845 0.78 PYCR1 (0.76) PYCR1MAPT
SCHEMBL13123456 0.77 SCN8A (0.50) SCN8AEPHX2NR1H4KDM1AHTR2C
SCHEMBL19690421 0.77 PYCR1 (0.59) PYCR1SCN8AALDH1A1
SCHEMBL3215494 0.77 ALDH1A1 (0.44) EPHX2NR1H4KDM1AHTR2CALDH1A1
SCHEMBL178527 0.77 EPHX2 (0.51) SCN8AEPHX2NR1H4KDM1AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2246329-A1 4(1H)-pyridinone derivatives and their use as antimalaria agents Glaxo Group Limited (GB) 2010-11-03 EP disclosed