SCHEMBL3394993

SCHEMBL3394993

CS(=O)(=O)c1ccc(CN2C(=O)NC3(CCN(CC4CN(C(=O)C5CCC(F)(F)CC5)CC4c4ccccc4)CC3)C2=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 18/20 0.46
KDM1A O60341 1/20 0.43
MAOB P27338 1/20 0.43
NR1H2 P55055 1/20 0.40
NR1H3 Q13133 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3394998 1.00 CCR5 (0.46) CCR5KDM1AMAOBNR1H2NR1H3
Hydrochloric Acid SCHEMBL3395052 0.99 CCR5 (0.45) CCR5KDM1AMAOBNR1H2NR1H3
Hydrochloric Acid SCHEMBL3395048 0.99 CCR5 (0.45) CCR5KDM1AMAOBNR1H2NR1H3
SCHEMBL3391654 0.95 CCR5 (0.49) CCR5KDM1AMAOB
SCHEMBL3391658 0.95 CCR5 (0.49) CCR5KDM1AMAOB
Hydrochloric Acid SCHEMBL3394503 0.94 CCR5 (0.48) CCR5KDM1AMAOB
Hydrochloric Acid SCHEMBL3394502 0.94 CCR5 (0.48) CCR5KDM1AMAOB
SCHEMBL3387158 0.93 CCR5 (0.54) CCR5KDM1AMAOB
SCHEMBL3387164 0.93 CCR5 (0.54) CCR5KDM1AMAOB
Hydrochloric Acid SCHEMBL3391810 0.93 CCR5 (0.53) CCR5KDM1AMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7709642-B2 Spirohydantoin compounds and methods for the modulation of chemokine receptor activity VIROCHEM PHARMA, INC. (CA) 2010-05-04 US claimed