Pyridine

Pyridine

SCHEMBL3395217

C[Si](C)(C)C(F)(C(=O)N(F)F)[Si](C)(C)C.c1ccncc1

nearest known ligand 0.33

Full drug profile on Sugi Atlas →

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.33
NAPRT Q6XQN6 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2851395 0.78
Dimethylformamide SCHEMBL3299693 0.73 TSHR (0.36) TSHR
Pyridine SCHEMBL5676908 0.72 TSHR (0.35) TSHRNAPRTTDP1
Pyridine SCHEMBL20661000 0.70 TSHR (0.33) TSHRNAPRTTDP1
Pyridine SCHEMBL28868409 0.69 NAPRT (0.45) TSHRNAPRTTDP1
Trifluoroacetic Acid SCHEMBL16824180 0.68 NAPRT (0.50) TSHRNAPRTTDP1
Trifluoroacetic Acid SCHEMBL158703 0.68 NAPRT (0.50) TSHRNAPRTTDP1
Trifluoroacetic Acid SCHEMBL9068482 0.68 NAPRT (0.50) TSHRNAPRTTDP1
Oxalic Acid SCHEMBL5874777 0.67 NAPRT (0.64) TSHRNAPRTTDP1
Oxalic Acid SCHEMBL4224676 0.67 NAPRT (0.64) TSHRNAPRTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 47 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1576123-B1 PROCESS FOR THE BIOLOGICAL PRODUCTION OF 1,3-PROPANEDIOL WITH HIGH YIELD DU PONT (US) 2010-12-29 EP disclosed
US-7745184-B2 Using transgenic escherichia expressing galactose-proton symporter and reduced glycerolaldehyde 3-phosphate dehydrogenase as bioreactor for 1,3-propanediol production E. I. DU PONT DE NEMOURS AND CO. (US) 2010-06-29 US disclosed
EP-0942989-B1 METHOD FOR THE PRODUCTION OF 1,3-PROPANEDIOL BY RECOMBINANT ORGANISMS DU PONT (US) 2009-12-23 EP disclosed
US-7629161-B2 Bioconversion of a fermentable carbon source to 1,3-propanediol by a single microorganism E.I. DU PONT DE NEMOURS AND COMPANY (US) 2009-12-08 US disclosed
US-20090253192-A1 PROCESS FOR THE BIOLOGICAL PRODUCTION OF 1,3-PROPANEDIOL WITH HIGH TITER E. I. DU PONT DE NEMOURS AND COMPANY (US) 2009-10-08 US disclosed
US-7582457-B2 Method for the production of 1,3-propanediol by recombinant organisms comprising genes for coenzyme B12 synthesis E.I. DU PONT DE NEMOURS AND COMPANY (US) 2009-09-01 US disclosed
US-7504250-B2 Process for the biological production of 1,3-propanediol with high titer E. I. DU PONT DE NEMOURS AND COMPANY (US) 2009-03-17 US disclosed
EP-0826057-B1 BIOCONVERSION OF A FERMENTABLE CARBON SOURCE TO 1,3-PROPANEDIOL BY A SINGLE MICROORGANISM DU PONT (US) 2009-01-21 EP disclosed
US-7452710-B2 Process for the biological production of 1,3-propanediol with high titer E.I. DU PONT DE NEMOURS AND COMPANY (US) 2008-11-18 US disclosed
EP-1076708-B1 METHOD FOR THE PRODUCTION OF 1,3-PROPANEDIOL BY RECOMBINANT ORGANISMS COMPRISING GENES FOR VITAMIN B 12 TRANSPORT DU PONT (US) 2008-10-08 EP disclosed
EP-1076708-A2 METHOD FOR THE PRODUCTION OF 1,3-PROPANEDIOL BY RECOMBINANT ORGANISMS COMPRISING GENES FOR VITAMIN B 12 TRANSPORT E.I. DU PONT DE NEMOURS AND COMPANY (US) 2001-02-21 EP disclosed
US-6171836-B1 EXPRESSION CASSETTE INCLUDING REGULATORY SEQUENCES AND HETEROLOGOUS DNA ENCODING TWO OR MORE ENZYMES FROM METABOLIC PATHWAY FOR BIOCONVERSTION OF CHOLESTEROL TO HYDROCORTISONE; FOR RECOMBINANT PRODUCTION HOECHST MARION ROUSSEL (FR) 2001-01-09 US disclosed
US-6136576-A EFFICIENT PRODUCTION BY CULTURING A RECOMBINANT MICROORGANISM HAVING AT LEAST NUCLEIC ACIDS ENCODING A DEHYDRATASE AND PROTEIN X IN PRESENCE OF AT LEAST ONE CARBON SOURCE GENENCOR INTERNATIONAL, INC. (US) 2000-10-24 US disclosed
US-6013494-A USING ENZYMES CODED IN EXPRESSION VECTORS TO MAKE A PROPANEDIOL; CULTURING TRANSFORMED MICROORGANISM IN THE PRESENCE OF MONOSACCARIDES, OLIGIOSACCHARIDES, AND POLYSACCHARIDES, RECOVERING THE 1,3-PROPANEDIOL E. I. DU PONT DE NEMOURS AND COMPANY (US) 2000-01-11 US disclosed
WO-1999058686-A2 METHOD FOR THE PRODUCTION OF 1,3-PROPANEDIOL BY RECOMBINANT ORGANISMS COMPRISING GENES FOR VITAMIN B12 TRANSPORT E.I. DU PONT DE NEMOURS AND COMPANY (US) 1999-11-18 WO disclosed
EP-0942989-A1 METHOD FOR THE PRODUCTION OF 1,3-PROPANEDIOL BY RECOMBINANT ORGANISMS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1999-09-22 EP disclosed
US-5869283-A ENCODING A PROTEIN, WHICH IS FUNCTIONAL, ALONE OR IN COOPERATION WITH ONE OR MORE ADDITIONAL PROTEINS, OF CATALYZING AN OXIDATION STEP IN THE BIOLOGICAL PATHWAY FOR CONVERSION OF CHOLESTEROL INTO HYDROCORTISONE ROUSSEL UCLAF (FR) 1999-02-09 US disclosed
WO-1998021339-A1 METHOD FOR THE PRODUCTION OF 1,3-PROPANEDIOL BY RECOMBINANT ORGANISMS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1998-05-22 WO disclosed
WO-1989010963-A1 PROCESS FOR THE BIOCHEMICAL OXIDATION OF STEROIDS AND GENETICALLY ENGINEERED CELLS TO BE USED THEREFOR GIST-BROCADES N.V. (NL) 1989-11-16 WO disclosed
EP-0340878-A1 Process for the biochemical oxidation of steroids and genetically engineered cells to be used therefor ROUSSEL UCLAF (FR) 1989-11-08 EP disclosed