SCHEMBL3395404

SCHEMBL3395404

Cc1cc(C#N)ccc1-c1nc(NCc2cc(-c3ccccc3)[nH]n2)ncc1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.47
ADORA2A P29274 2/20 0.38
ADORA2B P29275 2/20 0.38
ADORA1 P30542 2/20 0.38
TRIM33 Q9UPN9 1/20 0.37
GSK3A P49840 2/20 0.36
GSK3B P49841 2/20 0.36
CYP1A2 P05177 6/20 0.36
CYP3A4 P08684 5/20 0.36
CYP2C19 P33261 3/20 0.36
TSHR P16473 2/20 0.36
CYP2D6 P10635 2/20 0.36
CLK4 Q9HAZ1 6/20 0.36
ALDH1A1 P00352 4/20 0.36
HSD17B10 Q99714 3/20 0.36
MERTK Q12866 1/20 0.36
CCNB2 O95067 1/20 0.36
CDK1 P06493 1/20 0.36
CCNB1 P14635 1/20 0.36
RPS6KB1 P23443 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13425737 0.93 KCNH2 (0.46) KCNH2ADORA2AADORA2BADORA1TRIM33
SCHEMBL3434434 0.90 KCNH2 (0.40) KCNH2ADORA2AADORA2BADORA1TRIM33
SCHEMBL13425773 0.90 KCNH2 (0.43) KCNH2ADORA2AADORA2BADORA1TRIM33
SCHEMBL13425821 0.89 KCNH2 (0.41) KCNH2ADORA2AADORA2BADORA1TRIM33
SCHEMBL13425734 0.88 ADORA2B (0.48) ADORA2AADORA2BADORA1CYP1A2CYP3A4
SCHEMBL3394361 0.86 KDR (0.41) KCNH2CYP1A2CYP3A4CYP2C19TSHR
SCHEMBL13425543 0.86 NR1H4 (0.37) ADORA1CYP1A2CYP3A4CYP2C19TSHR
SCHEMBL13425809 0.85 KCNH2 (0.49) KCNH2GSK3AGSK3BCYP1A2CYP3A4
SCHEMBL13425775 0.83 GPR84 (0.38) ADORA1GSK3AGSK3BCCNB2CDK1
SCHEMBL13425741 0.82 KDR (0.37) ADORA2AADORA2BADORA1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed