SCHEMBL3397349

SCHEMBL3397349

OB(O)c1ccc(CN2CCC(c3ccc(OC(F)(F)F)cc3)CC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.52
TSHR P16473 1/20 0.52
BCHE P06276 4/20 0.51
ACHE P22303 4/20 0.51
BACE1 P56817 4/20 0.51
TEAD1 P28347 2/20 0.48
GRM2 Q14416 1/20 0.45
JAK2 O60674 1/20 0.45
JAK1 P23458 1/20 0.45
TYK2 P29597 1/20 0.45
JAK3 P52333 1/20 0.45
LMNA P02545 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
EPHX2 P34913 1/20 0.43
CHRM2 P08172 1/20 0.43
CHRM1 P11229 1/20 0.43
DRD4 P21917 3/20 0.43
DRD2 P14416 2/20 0.43
DRD3 P35462 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3398473 0.84 TEAD1 (0.57) ALDH1A1TSHRBCHEACHEBACE1
SCHEMBL12419665 0.79 MEN1 (0.60) ACHEMEN1KMT2ADRD4DRD2
SCHEMBL5542857 0.78 ALDH1A1 (0.64) ALDH1A1TSHRBCHEACHEBACE1
SCHEMBL12419666 0.77 MEN1 (0.50) ALDH1A1BCHEACHELMNAMEN1
SCHEMBL13070020 0.75 MBTD1 (0.51) ALDH1A1TSHRBCHEACHEBACE1
SCHEMBL2553332 0.75 KCNH2 (0.45) ALDH1A1BCHEACHEBACE1TEAD1
SCHEMBL15570990 0.75 KDM1A (0.40) JAK2JAK1TYK2JAK3DRD2
SCHEMBL19538689 0.75 TSHR (0.60) ALDH1A1TSHRBCHEACHEBACE1
SCHEMBL15591085 0.75 ALDH1A1 (0.68) ALDH1A1TSHRBCHEACHEBACE1
SCHEMBL2856132 0.75 ALDH1A1 (0.64) ALDH1A1TSHRBCHEACHEBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2246329-A1 4(1H)-pyridinone derivatives and their use as antimalaria agents Glaxo Group Limited (GB) 2010-11-03 EP disclosed