SCHEMBL3398247

SCHEMBL3398247

Cc1nc(-c2cc(Cl)ccc2Cl)sc1C(=O)NCCN1CCCC1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.48
DPP4 P27487 1/20 0.48
DPP8 Q6V1X1 1/20 0.48
CHRM4 P08173 1/20 0.48
PDE2A O00408 1/20 0.45
PDE10A Q9Y233 1/20 0.45
CNR1 P21554 1/20 0.45
DRD2 P14416 1/20 0.45
ABL1 P00519 2/20 0.44
GAA P10253 2/20 0.44
EPHX2 P34913 1/20 0.44
NPSR1 Q6W5P4 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3405826 0.99 DPP4 (0.49) ALDH1A1DPP4DPP8CHRM4PDE2A
SCHEMBL3404779 0.94 MAPK1 (0.49) ALDH1A1CHRM4DRD2GAANPSR1
SCHEMBL3402107 0.93 DRD2 (0.47) ALDH1A1CHRM4DRD2GAANPSR1
SCHEMBL3401355 0.92 DPP4 (0.54) ALDH1A1DPP4DPP8CHRM4PDE2A
SCHEMBL3400943 0.91 DPP4 (0.56) ALDH1A1DPP4DPP8CHRM4CNR1
SCHEMBL3402323 0.88 DPP4 (0.49) ALDH1A1DPP4DPP8CHRM4DRD2
SCHEMBL3402762 0.88 NPC1 (0.53) ALDH1A1CHRM4PDE2APDE10ANPSR1
SCHEMBL3405324 0.88 CHRM4 (0.51) ALDH1A1CHRM4PDE2APDE10AGAA
SCHEMBL3402094 0.87 DPP4 (0.50) ALDH1A1DPP4DPP8CHRM4DRD2
SCHEMBL3403391 0.87 CHRM4 (0.50) ALDH1A1CHRM4PDE2APDE10AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed