SCHEMBL3399083

SCHEMBL3399083

FC(F)(F)c1ccc(-c2ncc[nH]2)cc1.N#Cc1ccc(F)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.54
DGAT1 O75907 2/20 0.49
SOAT1 P35610 1/20 0.49
KCNH2 Q12809 1/20 0.49
GCGR P47871 2/20 0.46
MAPK14 Q16539 2/20 0.46
ALOX5 P09917 2/20 0.46
MAPK13 O15264 1/20 0.46
MAPK12 P53778 1/20 0.46
MAPK11 Q15759 1/20 0.46
NISCH Q9Y2I1 2/20 0.42
MTOR P42345 1/20 0.41
ADK P55263 1/20 0.41
CYP3A4 P08684 2/20 0.40
CYP3A5 P20815 1/20 0.40
CYP19A1 P11511 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL772274 0.83 NISCH (0.58) KIF11NISCHMTORADKCYP3A4
SCHEMBL378124 0.83 NISCH (0.58) KCNH2NISCHMTORADKCYP3A4
Hydrochloric Acid SCHEMBL29165675 0.81 NISCH (0.56) KCNH2NISCHMTORADKCYP3A4
SCHEMBL771236 0.78 NISCH (0.64) KCNH2GCGRMAPK14MAPK13MAPK12
Hydrochloric Acid SCHEMBL28346045 0.76 NISCH (0.62) KCNH2GCGRMAPK14MAPK13MAPK12
Bromide SCHEMBL28348957 0.76 NISCH (0.62) KCNH2GCGRMAPK14MAPK13MAPK12
SCHEMBL1507855 0.75 KIF11 (0.47) KIF11DGAT1SOAT1KCNH2CYP3A4
SCHEMBL13063632 0.73 KIF11 (1.00) KIF11DGAT1SOAT1KCNH2CYP3A4
SCHEMBL3456838 0.73 KIF11 (1.00) KIF11DGAT1SOAT1KCNH2CYP3A4
SCHEMBL29160561 0.72 NISCH (0.56) KCNH2GCGRMAPK14MAPK13MAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247603-A1 PESTICIDAL COMPOSITIONS Dow AgroSciences LLC (US) 2010-11-10 EP disclosed
WO-2009102736-A1 PESTICIDAL COMPOSITIONS DOW AGROSCIENCES LLC (US) 2009-08-20 WO disclosed