SCHEMBL3399230

SCHEMBL3399230

[CH2]c1cnn(-c2cccnc2)c1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.53
MTOR P42345 2/20 0.44
RPTOR Q8N122 1/20 0.42
MLST8 Q9BVC4 1/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2E1 P05181 2/20 0.41
GRM4 Q14833 1/20 0.40
HTT P42858 1/20 0.40
ELANE P08246 1/20 0.39
GAA P10253 1/20 0.39
EP300 Q09472 1/20 0.38
KAT2B Q92831 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNA4 P43681 1/20 0.38
CYP11B2 P19099 1/20 0.37
RIPK2 O43353 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12410587 0.81 CYP2A6 (0.56) CYP2A6MTORRPTORMLST8CYP3A4
SCHEMBL1304053 0.80 GAA (0.59) MTORGRM4HTTGAA
SCHEMBL12004826 0.79 CYP2A6 (0.55) CYP2A6MTORRPTORMLST8CYP3A4
SCHEMBL28194647 0.78 CYP2A6 (0.53) CYP2A6MTORRPTORMLST8CYP3A4
SCHEMBL2121774 0.78 CYP2A6 (0.53) CYP2A6MTORRPTORMLST8CYP3A4
SCHEMBL31132042 0.78 CYP2A6 (0.53) CYP2A6MTORRPTORMLST8CYP3A4
SCHEMBL3156531 0.78 CYP2A6 (0.53) CYP2A6MTORRPTORMLST8CYP3A4
SCHEMBL247216 0.78 CYP2A6 (0.53) CYP2A6MTORRPTORMLST8CYP3A4
SCHEMBL28195223 0.77 CYP2A6 (0.49) CYP2A6MTORRPTORMLST8CYP3A4
SCHEMBL12410440 0.76 CYP2A6 (0.54) CYP2A6MTORRPTORMLST8CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2233493-A1 Macrolides Pfizer Products Inc. (US) 2010-09-29 EP disclosed