SCHEMBL12410440

SCHEMBL12410440

c1cncc(-c2cnn(-c3cccnc3)c2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.54
ALDH1A1 P00352 3/20 0.54
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
L3MBTL1 Q9Y468 2/20 0.50
GRM4 Q14833 2/20 0.49
CHRNB2 P17787 1/20 0.45
CHRNA5 P30532 1/20 0.45
CHRNA4 P43681 1/20 0.45
RIPK2 O43353 3/20 0.44
DYRK1A Q13627 1/20 0.43
MTOR P42345 2/20 0.43
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
ALOX15 P16050 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12410587 0.94 CYP2A6 (0.56) CYP2A6ALDH1A1CYP1A2CYP3A4L3MBTL1
SCHEMBL12410565 0.88 MELK (0.54) CYP2A6CYP3A4GRM4RIPK2DYRK1A
SCHEMBL12482554 0.83 GRM4 (0.52) CYP2A6ALDH1A1CYP1A2CYP3A4L3MBTL1
SCHEMBL12410455 0.83 MAP4K4 (0.52) CYP2A6GRM4RIPK2MTOR
SCHEMBL29992360 0.83 MIF (0.61) CYP2A6ALDH1A1CYP1A2CYP3A4L3MBTL1
SCHEMBL16633967 0.83 MAPT (0.47) CYP2A6ALDH1A1CYP1A2CYP3A4L3MBTL1
SCHEMBL16634221 0.81 MKNK1 (0.56) CYP1A2CYP3A4GRM4TP53MAPT
SCHEMBL12410466 0.80 MAPKAPK2 (0.55) CYP2A6ALDH1A1CYP1A2CYP3A4GRM4
SCHEMBL12410456 0.80 GRM4 (0.47) CYP2A6CYP3A4GRM4
SCHEMBL12005171 0.80 PTGS2 (0.40) CYP2A6CYP3A4GRM4RIPK2ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9066518-B2 Heterocyclic compounds as pesticides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-06-30 US disclosed
US-9066518-B2 Heterocyclic compounds as pesticides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-06-30 US disclosed
EP-2488030-B1 1-(PYRID-3-YL)-PYRAZOLES AND 1-(PYRIMID-5-YL)-PYRAZOLES AS PEST CONTROLLERS BAYER CROPSCIENCE AG (DE) 2015-01-07 EP disclosed
US-20140221362-A1 Heterocyclic Compounds as Pesticides BAYER CROPSCIENCE AG (DE) 2014-08-07 US disclosed
US-20140221362-A1 Heterocyclic Compounds as Pesticides BAYER CROPSCIENCE AG (DE) 2014-08-07 US disclosed
US-20110166143-A1 Heterocyclic Compounds as Pesticides BAYER CROPSCIENCE AG (DE) 2011-07-07 US disclosed
US-20110166143-A1 Heterocyclic Compounds as Pesticides BAYER CROPSCIENCE AG (DE) 2011-07-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140221362-A1 Heterocyclic Compounds as Pesticides DDT, ACHE, BCHE CYP2A6 256/4885ALDH1A1 1595/4885CYP1A2 75/4885
US-20110166143-A1 Heterocyclic Compounds as Pesticides DDT, ACHE, BCHE CYP2A6 256/4885ALDH1A1 1595/4885CYP1A2 75/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.