SCHEMBL12410587

SCHEMBL12410587

c1cncc(-n2cc(-c3cnn(-c4cccnc4)c3)cn2)c1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.56
GRM4 Q14833 4/20 0.53
RIPK2 O43353 3/20 0.46
MTOR P42345 2/20 0.46
CYP3A4 P08684 2/20 0.44
MELK Q14680 2/20 0.44
HTR2B P41595 1/20 0.44
MTNR1A P48039 1/20 0.44
KCNH2 Q12809 1/20 0.44
RPTOR Q8N122 1/20 0.44
MLST8 Q9BVC4 1/20 0.44
ADORA2A P29274 1/20 0.44
ADORA2B P29275 1/20 0.44
ADORA1 P30542 1/20 0.44
CYP2E1 P05181 1/20 0.43
ALDH1A1 P00352 1/20 0.43
CYP1A2 P05177 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12410440 0.94 CYP2A6 (0.54) CYP2A6GRM4RIPK2MTORCYP3A4
SCHEMBL12410565 0.93 MELK (0.54) CYP2A6GRM4RIPK2MTORCYP3A4
SCHEMBL12410455 0.88 MAP4K4 (0.52) CYP2A6GRM4RIPK2MTORMELK
SCHEMBL12410466 0.84 MAPKAPK2 (0.55) CYP2A6GRM4CYP3A4KCNH2ALDH1A1
SCHEMBL12410456 0.84 GRM4 (0.47) CYP2A6GRM4CYP3A4MELKKCNH2
SCHEMBL3923984 0.84 GRM5 (0.60) CYP2A6GRM4RIPK2HTR2BMTNR1A
SCHEMBL2712276 0.83 MKNK1 (0.59) GRM4RIPK2MELKALDH1A1
SCHEMBL12004826 0.82 CYP2A6 (0.55) CYP2A6GRM4RIPK2MTORCYP3A4
SCHEMBL12410593 0.82 CYP2A6 (0.47) CYP2A6GRM4RIPK2MTORHTR2B
SCHEMBL12410547 0.81 CYP2A6 (0.58) CYP2A6GRM4RIPK2MTORHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9066518-B2 Heterocyclic compounds as pesticides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-06-30 US disclosed
US-9066518-B2 Heterocyclic compounds as pesticides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-06-30 US disclosed
EP-2488030-B1 1-(PYRID-3-YL)-PYRAZOLES AND 1-(PYRIMID-5-YL)-PYRAZOLES AS PEST CONTROLLERS BAYER CROPSCIENCE AG (DE) 2015-01-07 EP disclosed
US-20140221362-A1 Heterocyclic Compounds as Pesticides BAYER CROPSCIENCE AG (DE) 2014-08-07 US disclosed
US-20140221362-A1 Heterocyclic Compounds as Pesticides BAYER CROPSCIENCE AG (DE) 2014-08-07 US disclosed
US-20110166143-A1 Heterocyclic Compounds as Pesticides BAYER CROPSCIENCE AG (DE) 2011-07-07 US disclosed
US-20110166143-A1 Heterocyclic Compounds as Pesticides BAYER CROPSCIENCE AG (DE) 2011-07-07 US disclosed
WO-2011045224-A1 1- (PYRID-3-YL) -PYRAZOLE AND 1- (PYRIMID-5-YL) -PYRAZOLE AS PESTICIDE BAYER CROPSCIENCE AG (DE) 2011-04-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140221362-A1 Heterocyclic Compounds as Pesticides DDT, ACHE, BCHE CYP2A6 256/4885GRM4 1196/4885RIPK2 1635/4885
US-20110166143-A1 Heterocyclic Compounds as Pesticides DDT, ACHE, BCHE CYP2A6 256/4885GRM4 1196/4885RIPK2 1635/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.