SCHEMBL3399324

SCHEMBL3399324

CCN(CC)C(CCOc1ccc(-c2ccc3[nH]c4nccc(Cl)c4c3c2)cc1)C(CCN(C)C)Oc1ccc(-c2ccc3[nH]c4nccc(Cl)c4c3c2)cc1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 10/20 0.42
BRAF P15056 3/20 0.34
ACHE P22303 2/20 0.34
MAOA P21397 2/20 0.33
SLC6A4 P31645 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
UTS2R Q9UKP6 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL676066 0.81 ALK (0.53) ALKBRAFACHEMAOA
SCHEMBL675823 0.78 ALK (0.51) ALKACHEHRH3UTS2R
SCHEMBL3668987 0.71 ALK (0.61) ALK
SCHEMBL675708 0.69 ALK (0.68) ALK
SCHEMBL3727917 0.68 MAOA (0.44) ALKMAOAHRH3UTS2R
SCHEMBL676245 0.66 ALK (0.62) ALK
SCHEMBL3722596 0.65 HRH3 (0.40) ALKACHEHRH3UTS2R
SCHEMBL675901 0.65 ALK (0.50) ALKMAOA
SCHEMBL675900 0.65 ALK (0.50) ALKMAOA
SCHEMBL3399377 0.65 LSS (0.47) ACHEMAOAHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010025872-A2 ALFA-CARBOLINE INHIBITORS OF NPM-ALK, RET, AND BCR-ABL UNIVERSITA' DEGLI STUDI DI MILANO-BICOCCA (IT) 2010-03-11 WO disclosed