SCHEMBL3399342

SCHEMBL3399342

COc1cccc(OC)c1-c1nc(C)c(C(=O)NCCN2CCCC2)s1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.49
POLB P06746 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.47
ALDH1A1 P00352 2/20 0.47
RXFP1 Q9HBX9 1/20 0.47
DRD2 P14416 3/20 0.47
ALOX15 P16050 1/20 0.46
KDM4E B2RXH2 1/20 0.46
HSD17B10 Q99714 1/20 0.46
DRD4 P21917 2/20 0.45
POLR1A O95602 1/20 0.44
PARP1 P09874 1/20 0.44
HTR1A P08908 1/20 0.44
ADRA1A P35348 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13310019 0.87 SRC (0.47) POLBSMN1; SMN2ALDH1A1PARP1
SCHEMBL3402676 0.85 PARP1 (0.46) KMT2APOLBALDH1A1PARP1
SCHEMBL3402635 0.84 MEN1 (0.47) KMT2APOLBPARP1
SCHEMBL3405815 0.84 MAPT (0.52) POLBDRD2KDM4EDRD4
SCHEMBL3403888 0.84 MAPT (0.53) KMT2APOLBSMN1; SMN2RXFP1
SCHEMBL3399763 0.84 CHRM4 (0.51) KMT2APOLBDRD2KDM4EPOLR1A
SCHEMBL3405818 0.84 SMN1; SMN2 (0.46) KMT2APOLBSMN1; SMN2ALDH1A1ALOX15
SCHEMBL3398904 0.83 POLB (0.60) POLBALDH1A1KDM4EHSD17B10
SCHEMBL3398788 0.83 MAPT (0.48) KMT2APOLBSMN1; SMN2ALDH1A1RXFP1
SCHEMBL3404043 0.83 SMN1; SMN2 (0.60) KMT2APOLBSMN1; SMN2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed