SCHEMBL3399485

SCHEMBL3399485

CC1CN=C(c2ncccc2O)N1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 3/20 0.51
PDCD1 Q15116 2/20 0.41
CD274 Q9NZQ7 2/20 0.41
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 3/20 0.41
HPGD P15428 2/20 0.41
KMT2A Q03164 1/20 0.40
HSD17B10 Q99714 2/20 0.35
GLA P06280 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
EGLN1 Q9GZT9 1/20 0.35
ADRA2A P08913 4/20 0.35
ADRA2B P18089 2/20 0.35
ADRA2C P18825 2/20 0.35
MMP2 P08253 1/20 0.33
CHRM1 P11229 1/20 0.33
TSHR P16473 1/20 0.33
COMT P21964 1/20 0.33
ADRA1A P35348 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3403577 0.71 NISCH (0.51) NISCHKDM4E
SCHEMBL687180 0.70 KDM4E (0.55) ALDH1A1KDM4EHPGDKMT2AHSD17B10
SCHEMBL29769309 0.70 KDM4E (0.55) ALDH1A1KDM4EHPGDKMT2AHSD17B10
SCHEMBL14029048 0.69 NISCH (0.85) NISCHPDCD1CD274ADRA2AADRA2B
SCHEMBL10816996 0.68 NISCH (1.00) NISCHGAAADRA2AADRA2BADRA2C
SCHEMBL11133133 0.67 NISCH (0.81) NISCHPDCD1CD274ADRA2AADRA2B
SCHEMBL2573127 0.64 KDM4E (0.54) ALDH1A1KDM4EHPGDKMT2AHSD17B10
SCHEMBL30570543 0.64 KDM4E (0.54) ALDH1A1KDM4EHPGDKMT2AHSD17B10
SCHEMBL28897793 0.64 ALDH1A1 (0.50) ALDH1A1KDM4EHPGDKMT2AHSD17B10
SCHEMBL22815116 0.63 KDM4E (0.48) ALDH1A1KDM4EHPGDKMT2AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010018458-A2 PHENOL DERIVATIVES AND METHODS OF USE THEREOF CRYSTALGENOMICS, INC. (KR) 2010-02-18 WO claimed
WO-2010018458-A2 PHENOL DERIVATIVES AND METHODS OF USE THEREOF CRYSTALGENOMICS, INC. (KR) 2010-02-18 WO disclosed