SCHEMBL3400446

SCHEMBL3400446

Cc1cc(F)cc(-c2nc(C)c(C(=O)N3CCN(C(C)C)CC3)s2)c1Cl

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.44
CNR1 P21554 1/20 0.40
RORC P51449 1/20 0.38
THRA P10827 2/20 0.36
THRB P10828 2/20 0.36
CES2 O00748 1/20 0.36
CHRNA7 P36544 1/20 0.36
PARP1 P09874 2/20 0.36
HRH3 Q9Y5N1 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HSP90AA1 P07900 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
DYRK2 Q92630 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3406038 0.85 HTR2C (0.47) HTR2CCNR1THRATHRBCES2
SCHEMBL3407762 0.85 HTR2C (0.47) HTR2CCNR1THRATHRBCES2
SCHEMBL3402068 0.83 HTR2C (0.47) HTR2CCNR1THRATHRBCES2
SCHEMBL3405297 0.83 HTR2C (0.43) HTR2CCNR1THRATHRBMEN1
SCHEMBL3406010 0.83 CNR1 (0.49) HTR2CCNR1THRATHRBPARP1
SCHEMBL3396826 0.82 HTR2C (0.46) HTR2CCNR1CHRNA7PARP1HRH3
SCHEMBL3404209 0.82 HTR2C (0.49) HTR2CCNR1THRATHRBCES2
SCHEMBL3405067 0.81 HTR2C (0.47) HTR2CCNR1THRATHRBCES2
SCHEMBL3404163 0.81 HTR2C (0.47) HTR2CCNR1CES2CHRNA7HRH3
SCHEMBL3401691 0.80 HTR2C (0.45) HTR2CCNR1HRH3KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed