SCHEMBL3400988

SCHEMBL3400988

Cc1nc(-c2cc(C(F)(F)F)ccc2Cl)sc1C(=O)NCCC1CCCN1C

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 4/20 0.53
CHRM3 P20309 6/20 0.45
ACKR3 P25106 2/20 0.44
PPARA Q07869 2/20 0.42
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
PPARD Q03181 2/20 0.42
LCK P06239 1/20 0.42
CACNA1B Q00975 1/20 0.40
APBA1 Q02410 1/20 0.40
CRHR1 P34998 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3400900 0.89 CHRM4 (0.54) CHRM4CHRM3ACKR3PPARAPPARD
SCHEMBL3405198 0.86 CHRM4 (0.67) CHRM4CHRM3ACKR3PPARANPC1
SCHEMBL3405324 0.85 CHRM4 (0.51) CHRM4PPARANPC1ALDH1A1GAA
SCHEMBL3401222 0.85 CHRM4 (0.56) CHRM4CHRM3ACKR3PPARANPC1
SCHEMBL3405413 0.85 CHRM4 (0.53) CHRM4CHRM3ACKR3PPARANPC1
SCHEMBL13310232 0.85 CHRM4 (0.57) CHRM4CHRM3ACKR3PPARANPC1
SCHEMBL3403391 0.84 CHRM4 (0.50) CHRM4PPARANPC1ALDH1A1GAA
SCHEMBL3401105 0.84 CHRM4 (0.49) CHRM4PPARANPC1ALDH1A1GAA
SCHEMBL3405526 0.84 PPARD (0.53) CHRM4CHRM3ACKR3PPARANPC1
SCHEMBL3400884 0.84 CHRM4 (0.54) CHRM4CHRM3ACKR3PPARAPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed