SCHEMBL13310232

SCHEMBL13310232

Cc1nc(-c2cccc(C(F)(F)F)c2)sc1C(=O)NCCC1CCCN1C

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 4/20 0.57
ALDH1A1 P00352 2/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
PPARA Q07869 3/20 0.55
ACKR3 P25106 1/20 0.51
CHRM3 P20309 5/20 0.51
MEN1 O00255 2/20 0.48
MAPT P10636 2/20 0.48
KMT2A Q03164 2/20 0.48
GHSR Q92847 1/20 0.46
NPC1 O15118 1/20 0.46
GAA P10253 1/20 0.46
PPARD Q03181 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3405198 0.89 CHRM4 (0.67) CHRM4ALDH1A1PPARAACKR3CHRM3
SCHEMBL3398440 0.89 ACKR3 (0.51) CHRM4PPARAACKR3CHRM3NPC1
SCHEMBL3400075 0.87 ACKR3 (0.54) CHRM4ALDH1A1PPARAACKR3CHRM3
SCHEMBL3402412 0.86 ACKR3 (0.53) CHRM4PPARAACKR3NPC1PPARD
SCHEMBL3402209 0.85 ACKR3 (0.52) CHRM4ALDH1A1SMN1; SMN2PPARAACKR3
SCHEMBL3399976 0.85 ACKR3 (0.52) CHRM4ALDH1A1SMN1; SMN2PPARAACKR3
SCHEMBL3404196 0.85 ALDH1A1 (0.60) CHRM4ALDH1A1SMN1; SMN2PPARAMEN1
SCHEMBL3400988 0.85 CHRM4 (0.53) CHRM4ALDH1A1PPARAACKR3CHRM3
SCHEMBL3405413 0.85 CHRM4 (0.53) CHRM4ALDH1A1PPARAACKR3CHRM3
SCHEMBL3402424 0.85 ACKR3 (0.50) CHRM4PPARAACKR3NPC1PPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed