SCHEMBL3401042

SCHEMBL3401042

COc1ccc(C(=O)NC2COCCn3c2nc(-c2ccncn2)cc3=O)c(OC)n1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 17/20 0.39
CYP2D6 P10635 5/20 0.37
CYP1A2 P05177 4/20 0.36
CYP3A4 P08684 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CSNK2A2 P19784 1/20 0.35
CSNK2A1 P68400 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3402354 0.90 RAB9A (0.36) GSK3BCYP2D6CYP1A2MEN1KMT2A
SCHEMBL4387202 0.89 GSK3B (0.41) GSK3BCYP2D6CYP1A2CYP3A4MEN1
SCHEMBL4381292 0.88 GSK3B (0.41) GSK3BCYP2D6CYP1A2CYP3A4MEN1
SCHEMBL3659041 0.87 GSK3B (0.45) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL3654678 0.86 GSK3B (0.44) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL3402193 0.86 GSK3B (0.42) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL3402173 0.86 GSK3B (0.45) GSK3BCYP2D6CYP1A2
SCHEMBL3399343 0.85 GSK3B (0.47) GSK3BCYP2D6CYP1A2
SCHEMBL3399684 0.85 CRBN (0.42) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL927355 0.85 GSK3B (0.39) GSK3BCYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247598-A1 SUBSTITUTED HETEROARYLAMIDE OXAZEPINOPYRIMIDONE DERIVATIVES Sanofi-Aventis (FR) 2010-11-10 EP disclosed
WO-2009095787-A1 SUBSTITUTED HETEROARYLAMIDE OXAZEPINOPYRIMIDONE DERIVATIVES SANOFI-AVENTIS (FR) 2009-08-06 WO disclosed