SCHEMBL3401052

SCHEMBL3401052

COc1cc(C)sc1C(=O)N1CCC(Cc2ccccc2)CC1

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.65
CYP2C19 P33261 2/20 0.65
MAPK14 Q16539 2/20 0.65
MEN1 O00255 10/20 0.58
KMT2A Q03164 10/20 0.58
HTR2B P41595 1/20 0.56
APOBEC3A P31941 1/20 0.54
APOBEC3G Q9HC16 1/20 0.54
NPC1 O15118 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.52
POLB P06746 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3401138 0.83 CYP2C9 (0.58) CYP2C9CYP2C19MAPK14MEN1KMT2A
SCHEMBL7234983 0.79 CYP2C9 (1.00) CYP2C9CYP2C19MAPK14MEN1KMT2A
SCHEMBL7604997 0.79 CYP2C9 (0.77) CYP2C9CYP2C19MAPK14MEN1KMT2A
SCHEMBL5823073 0.79 CYP2C9 (0.77) CYP2C9CYP2C19MAPK14MEN1KMT2A
SCHEMBL7231606 0.78 CYP2C9 (0.69) CYP2C9CYP2C19MAPK14MEN1KMT2A
SCHEMBL7239766 0.78 CYP2C9 (0.65) CYP2C9CYP2C19MAPK14MEN1KMT2A
SCHEMBL5820252 0.76 CYP2C9 (0.77) CYP2C9CYP2C19MAPK14MEN1KMT2A
SCHEMBL7244230 0.76 MEN1 (0.69) CYP2C9CYP2C19MAPK14MEN1KMT2A
SCHEMBL4919897 0.76 CYP2C9 (0.57) CYP2C9CYP2C19MAPK14MEN1KMT2A
SCHEMBL7239929 0.76 MGLL (0.66) CYP2C9CYP2C19MAPK14MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247588-A2 FUSED HETEROCYCLIC DERIVATIVE AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2010-11-10 EP disclosed
WO-2009107850-A2 FUSED HETEROCYCLIC DERIVATIVE AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-09-03 WO disclosed