SCHEMBL3400850

SCHEMBL3400850

COc1ccc(-c2nc(C)c(C(=O)N3CCN(C4CCCC4)CC3)s2)c(OC)c1OC

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
ALDH1A1 P00352 2/20 0.44
HPGD P15428 1/20 0.44
HRH3 Q9Y5N1 2/20 0.43
PKM P14618 1/20 0.42
GAA P10253 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13071985 0.93 HTR2C (0.43) HTR2CNPC1RAB9AALDH1A1HPGD
SCHEMBL3401060 0.91 HTR2C (0.48) HTR2CALDH1A1HPGDHRH3
SCHEMBL3399981 0.91 HTR2C (0.48) HTR2CALDH1A1HPGDHRH3
SCHEMBL3402627 0.86 RAB9A (0.50) HTR2CNPC1RAB9AALDH1A1HPGD
SCHEMBL3405361 0.86 RAB9A (0.53) HTR2CNPC1RAB9AALDH1A1HPGD
SCHEMBL3400125 0.86 HTR2C (0.56) HTR2CNPC1RAB9AALDH1A1HPGD
SCHEMBL3405124 0.85 NPC1 (0.45) HTR2CNPC1RAB9AALDH1A1HPGD
SCHEMBL3402441 0.85 NPC1 (0.47) HTR2CNPC1RAB9AALDH1A1HPGD
SCHEMBL3398414 0.84 KMT2A (0.48) NPC1RAB9AALDH1A1HPGDHRH3
SCHEMBL13072012 0.84 HTR2C (0.47) HTR2CALDH1A1HPGDHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed