Moexipril

Moexipril

SCHEMBL34030

CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1Cc2cc(OC)c(OC)cc2C[C@H]1C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACE

The experimentally established mechanism targets of Moexipril. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ACE known ✓ P12821 15/20 1.00
PDE3A Q14432 1/20 1.00
ABCB11 O95342 2/20 0.80
LMNA P02545 1/20 0.64
SMN1; SMN2 Q16637 1/20 0.59
AGTR2 P50052 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Moexipril SCHEMBL6508276 1.00 ACE (1.00) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL29376544 1.00 ACE (1.00) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL683321 1.00 ACE (1.00) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL22175779 1.00 ACE (1.00) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL678818 1.00 ACE (1.00) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL5159178 0.99 ACE (0.98) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL40877 0.99 ACE (0.98) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL14660386 0.99 ACE (0.98) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL30903896 0.99 ACE (0.98) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL5386742 0.99 ACE (0.98) ACEPDE3AABCB11LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 16388 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12617809-B2 Cardioprotective lipid and method of use SIGNPATH PHARMA, INC. (US) 2026-05-05 US claimed
US-20260083968-A1 COMPOSITIONS, SYSTEMS, AND METHODS FOR TREATING CANCER USING TUMOR TREATING FIELDS (TTFIELDS) AND ACE INHIBITORS NOVOCURE GMBH (CH) 2026-03-26 US claimed
EP-4710928-A2 METHODS OF TREATING IGA NEPHROPATHY WITH ATRASENTAN Chinook Therapeutics, Inc. (US) 2026-03-18 EP claimed
EP-4691556-A2 HUMANIZED ANTI-ACTH ANTIBODIES AND USE THEREOF H. Lundbeck A/S (DK) 2026-02-11 EP claimed
EP-4684832-A2 POTASSIUM-BINDING AGENTS FOR TREATING HYPERTENSION AND HYPERKALEMIA Vifor (International) Ltd. (CH) 2026-01-28 EP claimed
US-20260021079-A1 NOX INHIBITORS FOR USE IN THE TREATMENT OF ALPORT SYNDROME CALLIDITAS THERAPEUTICS SUISSE SA (CH) 2026-01-22 US claimed
EP-4680248-A1 PRODUCTS OF MANUFACTURE AND THERAPEUTIC COMPOSITIONS FOR TREATING, AMELIORATING OR PREVENTING VIRAL INFECTIONS AND METHODS FOR MAKING AND USING THEM Topelia Aust Limited (ACN 652 771 670) (AU) 2026-01-21 EP claimed
US-12527767-B2 Eye drops to treat chemically induced corneal damage THE CURATORS OF THE UNIVERSITY OF MISSOURI (US) 2026-01-20 US claimed
EP-2916851-B1 POTASSIUM-BINDING AGENTS FOR TREATING HYPERTENSION AND HYPERKALEMIA VIFOR INT LTD (CH) 2025-12-17 EP claimed
EP-4076652-B1 A PHARMACEUTICALLY ACCEPTABLE SALT OF ATRASENTAN FOR USE IN A METHOD OF TREATING IGA NEPHROPATHY CHINOOK THERAPEUTICS INC (US) 2025-12-03 EP claimed
US-5651985-A DRUG IN TABLET FORM WITH POLYVINYLPYRROLIDONE AND METHACRYLIC ACID POLYMER BAYER AKTIENGESELLSCHAFT (DE) 1997-07-29 US claimed
WO-1997002032-A1 METHOD OF TREATING RENAL DISEASE USING AN ACE INHIBITOR AND AN AII ANTAGONIST MERCK & CO., INC. (US) 1997-01-23 WO claimed
WO-1996024372-A2 COMBINATION OF ANGIOTENSIN CONVERTING ENZYME INHIBITOR, SIDE-EFFECT-REDUCED AMOUNT OF ALDOSTERONE ANTAGONIST AND DIURETIC G.D. SEARLE & CO. (US) 1996-08-15 WO claimed
WO-1996024373-A2 COMBINATION OF ANGIOTENSIN CONVERTING ENZYME INHIBITOR AND SIDE-EFFECT-REDUCED AMOUNT OF ALDOSTERONE ANTAGONIST G.D. SEARLE & CO. (US) 1996-08-15 WO claimed
EP-0488059-B1 Use of a combination of an ace inhibitor with a calcium antagonist in the treatment of proteinuria HOECHST AG (DE) 1995-09-06 EP claimed
EP-0669129-A2 Expandable release controlled medicaments BAYER AG (DE) 1995-08-30 EP claimed
WO-1994028924-A1 COMBINATION OF ANGIOTENSIN CONVERTING ENZYME INHIBITORS AND AII ANTAGONISTS LABORATOIRES MERCK SHARP ET DOHME CHIBRET (FR) 1994-12-22 WO claimed
EP-0629408-A1 Combination of angiotensin converting enzyme inhibitors and AII antagonists LABORATOIRES MERCK, SHARP & DOHME-CHIBRET (FR) 1994-12-21 EP claimed
CN-1072601-A Angiotensin-convertion enzyme inhibitor and calcium antagonist are united and are used for the treatment of albuminuria HOECHST AG (DE) 1993-06-02 CN claimed
EP-0488059-A2 Use of a combination of an ace inhibitor with a calcium antagonist in the treatment of proteinuria HOECHST AKTIENGESELLSCHAFT (DE) 1992-06-03 EP claimed