Moexipril

Moexipril

SCHEMBL5159178

CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1Cc2cc(OC)c(OC)cc2C[C@H]1C(=O)O.[MgH2]

nearest known ligand 0.98

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACE

The experimentally established mechanism targets of Moexipril. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ACE known ✓ P12821 15/20 0.98
PDE3A Q14432 1/20 0.98
ABCB11 O95342 2/20 0.79
LMNA P02545 1/20 0.63
SMN1; SMN2 Q16637 1/20 0.58
AGTR2 P50052 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Moexipril SCHEMBL678818 0.99 ACE (1.00) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL683321 0.99 ACE (1.00) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL22175779 0.99 ACE (1.00) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL34030 0.99 ACE (1.00) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL29376544 0.99 ACE (1.00) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL6508276 0.99 ACE (1.00) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL14660386 0.98 ACE (0.98) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL40877 0.98 ACE (0.98) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL30903896 0.98 ACE (0.98) ACEPDE3AABCB11LMNASMN1; SMN2
Moexipril SCHEMBL5386742 0.98 ACE (0.98) ACEPDE3AABCB11LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1142878-B1 Pharmaceutical compositions comprising moexipril magnesium SHERMAN BERNARD CHARLES (CA) 2007-03-07 EP claimed
US-6767556-B2 HYPOTENSIVE AGENTS Sherman, Bernard Charles (CA) 2004-07-27 US claimed
US-20020037858-A1 Pharmaceutical compositions comprising moexipril magnesium APOTEX, INC. (CA) 2002-03-28 US claimed
EP-1142878-A2 Pharmaceutical compositions comprising moexipril magnesium SHERMAN, Bernard Charles (CA) 2001-10-10 EP claimed
EP-1142878-B1 Pharmaceutical compositions comprising moexipril magnesium SHERMAN BERNARD CHARLES (CA) 2007-03-07 EP disclosed
EP-1142878-B1 Pharmaceutical compositions comprising moexipril magnesium SHERMAN BERNARD CHARLES (CA) 2007-03-07 EP disclosed
WO-2005079772-A2 COMBINATION OF (S)-AMLODIPINE AND AN ACE INHIBITOR, AND METHODS FOR REDUCING HYPERTENSION SEPRACOR INC. (US) 2005-09-01 WO disclosed
US-6767556-B2 HYPOTENSIVE AGENTS Sherman, Bernard Charles (CA) 2004-07-27 US disclosed
US-6767556-B2 HYPOTENSIVE AGENTS Sherman, Bernard Charles (CA) 2004-07-27 US disclosed
US-6767556-B2 HYPOTENSIVE AGENTS Sherman, Bernard Charles (CA) 2004-07-27 US disclosed
EP-1142878-A3 Pharmaceutical compositions comprising moexipril magnesium SHERMAN, Bernard Charles (CA) 2003-09-17 EP disclosed
EP-1142878-A3 Pharmaceutical compositions comprising moexipril magnesium SHERMAN, Bernard Charles (CA) 2003-09-17 EP disclosed
US-20020037858-A1 Pharmaceutical compositions comprising moexipril magnesium APOTEX, INC. (CA) 2002-03-28 US disclosed
US-20020037858-A1 Pharmaceutical compositions comprising moexipril magnesium APOTEX, INC. (CA) 2002-03-28 US disclosed
US-20020037858-A1 Pharmaceutical compositions comprising moexipril magnesium APOTEX, INC. (CA) 2002-03-28 US disclosed
EP-1142878-A2 Pharmaceutical compositions comprising moexipril magnesium SHERMAN, Bernard Charles (CA) 2001-10-10 EP disclosed
EP-1142878-A2 Pharmaceutical compositions comprising moexipril magnesium SHERMAN, Bernard Charles (CA) 2001-10-10 EP disclosed
EP-1142878-A2 Pharmaceutical compositions comprising moexipril magnesium SHERMAN, Bernard Charles (CA) 2001-10-10 EP disclosed