SCHEMBL3403012

SCHEMBL3403012

Cc1nc(-c2ccc(C(F)(F)F)cc2)sc1C(=O)N1CCN(C(C)C)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.56
NPC1 O15118 1/20 0.56
GAA P10253 1/20 0.56
CNR1 P21554 1/20 0.52
EPHX2 P34913 2/20 0.50
PPARA Q07869 9/20 0.47
CHRM4 P08173 1/20 0.47
NR1H4 Q96RI1 1/20 0.46
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
HSP90AA1 P07900 1/20 0.46
MAPT P10636 1/20 0.46
CRHBP P24387 1/20 0.46
KMT2A Q03164 1/20 0.46
CRHR2 Q13324 1/20 0.46
PPARG P37231 3/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
PPARD Q03181 2/20 0.44
FFAR1 O14842 1/20 0.44
HTR2C P28335 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3399352 0.90 CNR1 (0.53) ALDH1A1NPC1GAACNR1PPARA
SCHEMBL3398823 0.89 ALDH1A1 (0.47) ALDH1A1NPC1GAACNR1EPHX2
SCHEMBL3399685 0.88 CNR1 (0.55) NPC1GAACNR1KDM4EMAPT
SCHEMBL3402418 0.88 ALDH1A1 (0.63) ALDH1A1NPC1GAACNR1EPHX2
SCHEMBL3405399 0.88 CNR1 (0.57) ALDH1A1NPC1GAACNR1KDM4E
SCHEMBL13071718 0.87 CNR1 (0.50) ALDH1A1NPC1GAACNR1PPARA
SCHEMBL3401410 0.86 EPHX2 (0.53) ALDH1A1NPC1GAACNR1EPHX2
SCHEMBL3405550 0.85 CNR1 (0.55) ALDH1A1NPC1GAACNR1KDM4E
SCHEMBL3401781 0.85 CNR1 (0.70) ALDH1A1NPC1GAACNR1MEN1
SCHEMBL3398840 0.84 CNR1 (0.54) NPC1GAACNR1KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed