SCHEMBL3403472

SCHEMBL3403472

CCCCc1ccc(-c2nc(C)c(C(=O)NCCC3CCCN3C)s2)cc1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 2/20 0.52
CHRM4 P08173 4/20 0.51
NPC1 O15118 1/20 0.45
HPGD P15428 1/20 0.45
PPARA Q07869 7/20 0.45
GLS O94925 1/20 0.44
PPARG P37231 2/20 0.42
PPARD Q03181 2/20 0.41
GAA P10253 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3405823 0.94 ACKR3 (0.53) ACKR3CHRM4NPC1HPGDPPARA
SCHEMBL3405398 0.91 ACKR3 (0.55) ACKR3CHRM4NPC1HPGDPPARA
SCHEMBL3399830 0.86 ACKR3 (0.54) ACKR3CHRM4NPC1HPGDPPARA
SCHEMBL3401785 0.86 ACKR3 (0.54) ACKR3CHRM4NPC1HPGDPPARA
SCHEMBL13310379 0.86 ACKR3 (0.50) ACKR3CHRM4NPC1HPGDPPARA
SCHEMBL3405220 0.85 ACKR3 (0.52) ACKR3CHRM4NPC1HPGDPPARA
SCHEMBL3403946 0.85 CHRM4 (0.56) ACKR3CHRM4NPC1HPGDPPARA
SCHEMBL3403598 0.85 ACKR3 (0.53) ACKR3CHRM4PPARAPPARGPPARD
SCHEMBL3398671 0.85 ACKR3 (0.53) ACKR3CHRM4NPC1HPGDPPARA
SCHEMBL3403460 0.85 CHRM4 (0.54) ACKR3CHRM4NPC1HPGDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed