SCHEMBL3404335

SCHEMBL3404335

CCN(CC)CCNC(=O)c1sc(-c2c(F)ccc(C)c2Cl)nc1C

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
HPGD P15428 2/20 0.42
GAA P10253 1/20 0.42
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 4/20 0.41
SMN1; SMN2 Q16637 4/20 0.41
KDM4E B2RXH2 3/20 0.41
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
POLB P06746 2/20 0.38
MCHR1 Q99705 1/20 0.38
LMNA P02545 1/20 0.38
ALOX15 P16050 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CHRM4 P08173 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3401216 0.87 GAA (0.41) MEN1KMT2AHPGDGAANPC1
SCHEMBL3401433 0.83 HTR2C (0.41) MEN1KMT2AGAANPC1ALDH1A1
SCHEMBL3399888 0.80 CHRM4 (0.45) KMT2AGAAALDH1A1MAPTNPSR1
SCHEMBL3404959 0.80 CHRM4 (0.44) GAAALDH1A1NPSR1LMNACHRM4
SCHEMBL3403957 0.78 PANK3 (0.46) TP53MEN1KMT2AHPGDGAA
SCHEMBL3398938 0.78 GAA (0.46) TP53MEN1KMT2AHPGDGAA
SCHEMBL3405341 0.78 KDM4E (0.51) TP53MEN1KMT2AHPGDGAA
SCHEMBL3399952 0.77 CHRM4 (0.55) CHRM4
SCHEMBL3399977 0.76 TSHR (0.53) TP53MEN1KMT2AHPGDGAA
SCHEMBL14545475 0.76 KDM4E (0.46) TP53MEN1KMT2AHPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed