SCHEMBL3404622

SCHEMBL3404622

COCCn1c(Cn2ccnc2-c2ncccc2F)nc2cnccc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.38
RAB9A P51151 2/20 0.38
KMT2A Q03164 2/20 0.38
TP53 P04637 2/20 0.38
NPC1 O15118 1/20 0.38
RPS6KA5 O75582 2/20 0.38
GRM2 Q14416 2/20 0.37
BRD4 O60885 2/20 0.36
MAPK14 Q16539 1/20 0.36
CYP1A2 P05177 3/20 0.34
CYP3A4 P08684 3/20 0.34
HSD17B10 Q99714 2/20 0.34
HPGD P15428 1/20 0.34
USP2 O75604 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GLA P06280 1/20 0.34
CYP2C19 P33261 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
GLP1R P43220 2/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3061412 0.88 RPS6KA5 (0.48) RAB9AKMT2ANPC1RPS6KA5GRM2
SCHEMBL3068284 0.86 RAB9A (0.39) TSHRRAB9AKMT2ATP53NPC1
SCHEMBL3055367 0.80 RPS6KA5 (0.40) RAB9AKMT2ANPC1RPS6KA5GRM2
SCHEMBL3064975 0.78 BRD4 (0.39) KMT2ATP53RPS6KA5GRM2BRD4
SCHEMBL3060221 0.76 CYP11B1 (0.38) RAB9AKMT2ANPC1RPS6KA5GRM2
SCHEMBL3062897 0.75 PKM (0.36) GRM2BRD4CYP1A2CYP2C19LMNA
SCHEMBL3068770 0.75 RPS6KA5 (0.45) RAB9AKMT2ANPC1RPS6KA5GRM2
SCHEMBL3060407 0.75 RPS6KA5 (0.37) RAB9AKMT2ATP53NPC1RPS6KA5
SCHEMBL3060473 0.74 PKM (0.41) TSHRRAB9ANPC1RPS6KA5BRD4
SCHEMBL3066024 0.74 RPS6KA5 (0.41) RAB9AKMT2ARPS6KA5HSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1368342-B3 BENZIMIDAZOLE AND PYRIDYLIMIDAZOLE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS NEUROGEN CORP (US) 2010-12-01 EP disclosed