SCHEMBL3404764

SCHEMBL3404764

Nc1ccc(C2CNCCO2)cc1

nearest known ligand 0.58

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.53
DRD3 P35462 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL82902 1.00 DRD2 (0.53) DRD2DRD3
SCHEMBL12695816 1.00 DRD2 (0.53) DRD2DRD3
Hydrochloric Acid SCHEMBL13505422 0.98 DRD2 (0.51) DRD2DRD3
Hydrochloric Acid SCHEMBL83201 0.98 DRD2 (0.51) DRD2DRD3
SCHEMBL503006 0.83 DRD2 (0.54) DRD2DRD3
SCHEMBL134338 0.83 DRD2 (0.54) DRD2DRD3
SCHEMBL503067 0.83 DRD2 (0.54) DRD2DRD3
SCHEMBL18290968 0.82 DRD2 (0.57) DRD2DRD3
SCHEMBL4249668 0.82 DRD2 (0.57) DRD2DRD3
SCHEMBL4242930 0.82 DRD2 (0.57) DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 203 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119591550-A Preparation method of molatinib and key intermediate 沈阳药科大学 2025-03-11 CN claimed
CN-114761406-B Hydropyrido [1,2-a ] pyrazine compounds for the treatment of autoimmune diseases 豪夫迈·罗氏有限公司 2024-04-19 CN claimed
EP-4069693-B1 HYDROPYRIDO[1,2-ALPHA]PYRAZINE COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE DISEASES HOFFMANN LA ROCHE (CH) 2024-03-20 EP claimed
US-11697636-B2 Substituted benzamides HOFFMANN-LA ROCHE INC. (US) 2023-07-11 US claimed
US-20230022297-A1 HYDROPYRIDO[1,2-a]PYRAZINE COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE DISEASE HOFFMANN-LA ROCHE INC. (US) 2023-01-26 US claimed
CN-114761406-A Hydropyrido [1,2-a ] pyrazine compounds for the treatment of autoimmune diseases 豪夫迈·罗氏有限公司 2022-07-15 CN claimed
EP-3187490-B1 SUBSTITUTED BENZAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2022-04-06 EP claimed
WO-2021110614-A1 HYDROPYRIDO[1,2-α]PYRAZINE COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE DISEASE F. HOFFMANN-LA ROCHE AG (CH) 2021-06-10 WO claimed
US-20210061760-A1 SUBSTITUTED BENZAMIDES HOFFMANN LA ROCHE (US) 2021-03-04 US claimed
CN-105793430-B Process for the preparation of chiral 2-arylmorpholines 豪夫迈·罗氏有限公司 2020-03-03 CN claimed
EP-3080284-A1 PROCESS FOR THE PREPARATION OF CHIRAL 2-ARYL MORPHOLINES F. Hoffmann-La Roche AG (CH) 2016-10-19 EP claimed
CN-106008533-A Cdk inhibitors G1治疗公司 2016-10-12 CN claimed
US-20160289718-A1 PROCESS FOR THE PREPARATION OF CHIRAL 2-ARYL MORPHOLINES HOFFMANN-LA ROCHE INC. (US) 2016-10-06 US claimed
US-9452980-B2 Substituted benzamides HOFFMANN-LA ROCHE INC. (US) 2016-09-27 US claimed
CN-105793430-A Process for the preparation of chiral 2-aryl morpholines 豪夫迈·罗氏有限公司 2016-07-20 CN claimed
CN-102648217-B Low molecular weight polymers of multifunctional multiple graft monomers CASTROL LTD. (GB) 2015-11-25 CN claimed
WO-2015086495-A1 PROCESS FOR THE PREPARATION OF CHIRAL 2-ARYL MORPHOLINES F. HOFFMANN-LA ROCHE AG (CH) 2015-06-18 WO claimed
EP-2516392-A1 SUBSTITUTED BENZAMIDE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2012-10-31 EP claimed
EP-0697036-A1 SILVER-CORROSION PROTECTION AGENT (II) Henkel Kommanditgesellschaft auf Aktien (DE) 1996-02-21 EP claimed
WO-1994026860-A1 SILVER-CORROSION PROTECTION AGENT (II) HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 1994-11-24 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230022297-A1 HYDROPYRIDO[1,2-a]PYRAZINE COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE DISEASE TLR7, TLR9, TLR5 DRD2 1892/4885DRD3 2400/4885
US-20160289718-A1 PROCESS FOR THE PREPARATION OF CHIRAL 2-ARYL MORPHOLINES TAAR1, TAAR5, TACR2 DRD2 182/4885DRD3 323/4885
US-20210061760-A1 SUBSTITUTED BENZAMIDES TAAR1, TAAR5, NPY1R DRD2 596/4885DRD3 1047/4885
US-11697636-B2 Substituted benzamides TAAR1, TAAR5, NPY1R DRD2 596/4885DRD3 1047/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.