SCHEMBL3404795

SCHEMBL3404795

Cc1cccc(-c2nc(C)c(C(=O)N3CCN(C4CCCC4)CC3)s2)c1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.53
HTR2C P28335 7/20 0.48
ALDH1A1 P00352 1/20 0.47
HPGD P15428 1/20 0.47
THRA P10827 2/20 0.47
THRB P10828 2/20 0.47
HRH3 Q9Y5N1 2/20 0.47
LMNA P02545 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
KMT2A Q03164 2/20 0.44
RAB9A P51151 2/20 0.44
MEN1 O00255 1/20 0.44
OXTR P30559 1/20 0.43
KDM2B Q8NHM5 1/20 0.42
NPC1 O15118 1/20 0.42
PKM P14618 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13309716 0.91 HRH3 (0.56) CNR1HTR2CTHRATHRBHRH3
SCHEMBL3405666 0.91 HRH3 (0.56) CNR1HTR2CTHRATHRBHRH3
SCHEMBL3405417 0.90 KMT2A (0.57) CNR1HTR2CALDH1A1HPGDTHRA
SCHEMBL3398926 0.90 TRPM8 (0.54) CNR1HTR2CALDH1A1HPGDTHRA
SCHEMBL3405619 0.89 CNR1 (0.48) CNR1HTR2CALDH1A1HPGDTHRA
SCHEMBL3400921 0.89 CNR1 (0.66) CNR1HTR2CALDH1A1HPGDHRH3
SCHEMBL3398454 0.89 MAPK1 (0.51) CNR1HTR2CALDH1A1HPGDTHRA
SCHEMBL3401828 0.89 HRH3 (0.52) CNR1HTR2CALDH1A1HPGDTHRA
SCHEMBL3403007 0.88 CNR1 (0.52) CNR1HTR2CALDH1A1HPGDTHRA
SCHEMBL3404810 0.88 CNR1 (0.49) CNR1HTR2CALDH1A1HPGDTHRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed