SCHEMBL3404822

SCHEMBL3404822

Cc1ccc(-c2nc(C)c(C(=O)N3CCN(C4CCCC4)CC3)s2)cc1C

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
THRA P10827 2/20 0.50
THRB P10828 2/20 0.50
KMT2A Q03164 2/20 0.48
CNR1 P21554 1/20 0.48
ALDH1A1 P00352 1/20 0.48
HPGD P15428 1/20 0.48
LMNA P02545 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HTR2C P28335 5/20 0.44
HRH3 Q9Y5N1 2/20 0.43
MEN1 O00255 1/20 0.43
RAB9A P51151 1/20 0.43
OXTR P30559 1/20 0.42
L3MBTL3 Q96JM7 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
KDM4E B2RXH2 1/20 0.41
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3405608 0.91 THRA (0.48) THRATHRBKMT2ACNR1ALDH1A1
SCHEMBL13071966 0.91 THRA (0.48) THRATHRBKMT2ACNR1ALDH1A1
SCHEMBL3403558 0.91 THRA (0.54) THRATHRBCNR1LMNAHTR2C
SCHEMBL3404539 0.91 THRA (0.54) THRATHRBCNR1LMNAHTR2C
SCHEMBL3405038 0.89 RAB9A (0.47) THRATHRBKMT2ACNR1ALDH1A1
SCHEMBL3403718 0.88 CNR1 (0.54) THRATHRBCNR1ALDH1A1HPGD
SCHEMBL3399794 0.88 THRA (0.49) THRATHRBCNR1ALDH1A1HPGD
SCHEMBL3405797 0.88 CNR1 (0.52) THRATHRBCNR1ALDH1A1HPGD
SCHEMBL3399902 0.88 THRA (0.49) THRATHRBCNR1ALDH1A1HPGD
SCHEMBL3399702 0.87 THRA (0.47) THRATHRBCNR1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed