SCHEMBL3405100

SCHEMBL3405100

C=CC(=O)NCc1ccc(F)c(-c2cccc(CN3CCN[C@@H](C)C3)c2)c1

nearest known ligand 0.72

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 19/20 0.72
CHRM2 P08172 6/20 0.72
CHRM1 P11229 6/20 0.72
KCNH2 Q12809 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4968514 0.87 CHRM3 (0.93) CHRM3CHRM2CHRM1KCNH2
SCHEMBL4099839 0.86 CHRM3 (0.86) CHRM3CHRM2CHRM1KCNH2
SCHEMBL3399242 0.85 CHRM3 (0.54) CHRM3CHRM2CHRM1KCNH2
SCHEMBL4095861 0.84 CHRM3 (0.88) CHRM3CHRM2CHRM1KCNH2
SCHEMBL4105534 0.84 CHRM3 (1.00) CHRM3CHRM2CHRM1KCNH2
SCHEMBL12725271 0.84 CHRM3 (1.00) CHRM3CHRM2CHRM1KCNH2
SCHEMBL12725342 0.83 CHRM3 (1.00) CHRM3CHRM2CHRM1KCNH2
SCHEMBL4108965 0.83 CHRM3 (0.85) CHRM3CHRM2CHRM1KCNH2
Trifluoroacetic Acid SCHEMBL4098300 0.83 CHRM3 (0.80) CHRM3CHRM2CHRM1KCNH2
SCHEMBL4106075 0.83 CHRM3 (0.85) CHRM3CHRM2CHRM1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2249646-A1 DUAL PHARMACOPHORES - PDE4-MUSCARINIC ANTAGONISTICS Glaxo Group Limited (GB) 2010-11-17 EP claimed
WO-2009100169-A1 DUAL PHARMACOPHORES - PDE4-MUSCARINIC ANTAGONISTICS GLAXO GROUP LIMITED (GB) 2009-08-13 WO claimed