SCHEMBL3405249

SCHEMBL3405249

Cc1nc(-c2cc(C(F)(F)F)cc(C(F)(F)F)c2)sc1C(=O)NCCN1CCCC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 2/20 0.53
ALDH1A1 P00352 2/20 0.50
NPC1 O15118 1/20 0.50
GAA P10253 1/20 0.50
CHRNB2 P17787 1/20 0.49
CHRNB4 P30926 1/20 0.49
CHRNA3 P32297 1/20 0.49
CHRNA4 P43681 1/20 0.49
PPARD Q03181 3/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
PPARA Q07869 10/20 0.47
EPHX2 P34913 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
PPARG P37231 3/20 0.44
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3403031 0.93 CHRM4 (0.51) CHRM4ALDH1A1NPC1GAACHRNB2
SCHEMBL3404196 0.90 ALDH1A1 (0.60) CHRM4ALDH1A1NPC1GAACHRNB2
SCHEMBL3403462 0.90 CHRM4 (0.65) CHRM4ALDH1A1NPC1GAACHRNB2
SCHEMBL3396893 0.86 SCN9A (0.48) CHRM4ALDH1A1NPC1GAAMEN1
SCHEMBL3405210 0.84 CHRM4 (0.51) CHRM4ALDH1A1NPC1GAAPPARA
SCHEMBL3403850 0.84 ALDH1A1 (0.57) CHRM4ALDH1A1NPC1GAAPPARD
SCHEMBL3405545 0.83 CHRM4 (0.50) CHRM4ALDH1A1NPC1GAAPPARA
SCHEMBL3399440 0.83 CHRM4 (0.62) CHRM4ALDH1A1NPC1GAACHRNB2
SCHEMBL3405324 0.83 CHRM4 (0.51) CHRM4ALDH1A1NPC1GAACHRNB2
SCHEMBL3405042 0.82 CHRM4 (0.49) CHRM4ALDH1A1NPC1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed