SCHEMBL3405546

SCHEMBL3405546

Cc1nc(-c2cccc(OC(C)C)c2)sc1C(=O)NCCN1CCCCC1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MKNK2 Q9HBH9 1/20 0.46
NPC1 O15118 2/20 0.45
HPGD P15428 2/20 0.45
ROCK1 Q13464 2/20 0.44
SCN9A Q15858 1/20 0.44
MAPT P10636 3/20 0.43
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
CHRM4 P08173 1/20 0.43
RAD52 P43351 1/20 0.43
GRK5 P34947 1/20 0.43
GSK3A P49840 1/20 0.43
GSK3B P49841 1/20 0.43
AVPR1B P47901 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
POLB P06746 1/20 0.42
GAA P10253 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3399919 0.99 HPGD (0.46) MKNK2NPC1HPGDROCK1SCN9A
SCHEMBL3405815 0.91 MAPT (0.52) NPC1HPGDROCK1MAPTKDM4E
SCHEMBL3429141 0.89 GLA (0.50) NPC1HPGDSCN9AMAPTKDM4E
SCHEMBL3429158 0.88 GLA (0.51) NPC1HPGDSCN9AMAPTKDM4E
SCHEMBL3399733 0.88 GLS (0.48) NPC1HPGDSCN9AMAPTALDH1A1
SCHEMBL3398475 0.86 PPARA (0.49) NPC1HPGDSCN9AMAPTALDH1A1
SCHEMBL3403919 0.85 ACKR3 (0.51) NPC1HPGDROCK1MAPTCHRM4
SCHEMBL3405410 0.83 HPGD (0.47) NPC1HPGDSCN9AMAPTKDM4E
SCHEMBL3398806 0.83 CHRM4 (0.54) NPC1HPGDSCN9AMAPTALDH1A1
SCHEMBL3400541 0.83 HPGD (0.48) NPC1HPGDMAPTALDH1A1CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed