SCHEMBL3405573

SCHEMBL3405573

Cc1cccc(C)c1-c1nc(C)c(C(=O)N2CCN(C(C)C)CC2)s1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.52
CNR1 P21554 1/20 0.50
PARP1 P09874 1/20 0.44
CES2 O00748 1/20 0.40
BCHE P06276 1/20 0.40
ACHE P22303 1/20 0.40
SIGLEC9 Q9Y336 1/20 0.39
HRH3 Q9Y5N1 3/20 0.39
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
MEN1 O00255 2/20 0.39
ALDH1A1 P00352 2/20 0.39
MAPT P10636 2/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HSP90AA1 P07900 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
KCNH2 Q12809 1/20 0.39
NPC1 O15118 1/20 0.39
NR1I2 O75469 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3404035 0.88 HTR2C (0.50) HTR2CCNR1PARP1CES2SIGLEC9
SCHEMBL3405446 0.88 CNR1 (0.47) HTR2CCNR1PARP1HRH3MEN1
SCHEMBL3400778 0.87 HTR2C (0.57) HTR2CCNR1PARP1CES2BCHE
SCHEMBL13309912 0.87 HTR2C (0.59) HTR2CCNR1PARP1CES2SIGLEC9
SCHEMBL3402656 0.86 HTR2C (0.48) HTR2CCNR1PARP1HRH3MEN1
SCHEMBL3401781 0.84 CNR1 (0.70) HTR2CCNR1PARP1HRH3MEN1
SCHEMBL3401181 0.84 CNR1 (0.47) HTR2CCNR1PARP1CES2SIGLEC9
SCHEMBL3399805 0.83 CNR1 (0.56) HTR2CCNR1PARP1HRH3ALDH1A1
SCHEMBL3405399 0.82 CNR1 (0.57) HTR2CCNR1PARP1HRH3ALDH1A1
SCHEMBL3405384 0.82 HTR2C (0.62) HTR2CCNR1PARP1CES2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8758976-B2 Positive photosensitive polyimide composition LG CHEM LTD. (KR) 2014-06-24 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed