SCHEMBL3405834

SCHEMBL3405834

CC(C)Oc1ccnc2ccc(C=C3SC(N)=CC3=O)nc12

nearest known ligand 0.32

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.32
GRIN3B O60391 1/20 0.31
GRIN1 Q05586 1/20 0.31
GRIN2C Q14957 1/20 0.31
CCNT1 O60563 1/20 0.30
CCNA2 P20248 1/20 0.30
CDK2 P24941 1/20 0.30
CDK9 P50750 1/20 0.30
CCNA1 P78396 1/20 0.30
CDK5 Q00535 1/20 0.30
CDK5R1 Q15078 1/20 0.30
IRAK4 Q9NWZ3 2/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
HPGD P15428 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3372661 0.84 MAPT (0.44) CDK9CDK5ALDH1A1MAPTHPGD
SCHEMBL3375305 0.84 MAPT (0.44) CDK9CDK5ALDH1A1MAPTHPGD
SCHEMBL3371078 0.76 CCR1 (0.41) MCHR1GRIN3BGRIN1GRIN2CCCNT1
SCHEMBL3373060 0.75 MAPT (0.35) GRIN3BGRIN1GRIN2CALDH1A1MAPT
SCHEMBL27718867 0.72 IRAK4 (0.32) GRIN3BGRIN1GRIN2CIRAK4
SCHEMBL3371468 0.72 KDM4E (0.34) ALDH1A1MAPTHPGD
SCHEMBL3370325 0.70 ALDH1A1 (0.34) CCNT1CCNA2CDK2CDK9CDK5
SCHEMBL3374050 0.70 ALDH1A1 (0.36) ALDH1A1MAPTHPGDSMN1; SMN2
SCHEMBL14337697 0.70 MKNK2 (0.35) ALDH1A1MAPTHPGDSMN1; SMN2
SCHEMBL3375285 0.70 ALDH1A1 (0.36) ALDH1A1MAPTHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1869036-B1 SUBSTITUTED 1,5-NAPHTHYRIDINE AZOLIDINONES AS CDK INHIBITORS HOFFMANN LA ROCHE (CH) 2010-11-03 EP disclosed