SCHEMBL3406434

SCHEMBL3406434

COc1cc(Nc2nccc(Cc3cc(F)c(F)c(F)c3)n2)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 14/20 0.39
CCNT1 O60563 9/20 0.39
PARP1 P09874 1/20 0.39
KDR P35968 1/20 0.39
CDK2 P24941 7/20 0.36
CCNA2 P20248 1/20 0.36
IGF1R P08069 2/20 0.36
BRD4 O60885 1/20 0.36
RET P07949 1/20 0.36
KCNH2 Q12809 1/20 0.36
AURKA O14965 1/20 0.36
AURKB Q96GD4 1/20 0.36
CCNE1 P24864 2/20 0.35
CCNE2 O96020 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3411154 0.88 PSEN1 (0.43) CDK9CCNT1CDK2IGF1RRET
SCHEMBL3409536 0.85 RET (0.40) CDK9CCNT1PARP1KDRCDK2
SCHEMBL3409757 0.84 CDK9 (0.47) CDK9CCNT1CDK2CCNA2BRD4
SCHEMBL3410466 0.84 PSEN1 (0.43) CDK9CCNT1CDK2IGF1RRET
SCHEMBL3408509 0.82 CDK9 (0.40) CDK9CCNT1PARP1KDRCDK2
SCHEMBL3412794 0.81 SYK (0.39) CDK9CCNT1CDK2CCNA2RET
SCHEMBL3410131 0.80 CCNA2 (0.37) CDK9CCNT1KDRCDK2CCNA2
SCHEMBL3412591 0.79 CDK9 (0.42) CDK9CCNT1PARP1KDRCDK2
SCHEMBL3406878 0.79 SYK (0.50)
SCHEMBL3406106 0.79 IGF1R (0.41) CDK9CCNT1PARP1KDRCDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed