SCHEMBL3407188

SCHEMBL3407188

NC(=O)c1cnc(-c2ncc(C(N)=O)cn2)nc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NNMT P40261 7/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
L3MBTL1 Q9Y468 2/20 0.45
KDM4E B2RXH2 1/20 0.45
F7 P08709 1/20 0.44
F3 P13726 1/20 0.44
SARM1 Q6SZW1 1/20 0.44
SIRT2 Q8IXJ6 1/20 0.44
SIRT6 Q8N6T7 1/20 0.44
SIRT1 Q96EB6 1/20 0.44
SIRT3 Q9NTG7 1/20 0.44
SIRT5 Q9NXA8 1/20 0.44
SIRT4 Q9Y6E7 1/20 0.44
TSHR P16473 2/20 0.43
POLB P06746 1/20 0.43
CYP3A4 P08684 1/20 0.43
PARP1 P09874 1/20 0.43
MAPT P10636 1/20 0.43
CYP2C19 P33261 1/20 0.43
RECQL P46063 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3407187 0.90 NNMT (0.48) NNMTSMN1; SMN2L3MBTL1KDM4EF7
SCHEMBL3141529 0.83 NNMT (0.58) NNMTSMN1; SMN2L3MBTL1KDM4EF7
SCHEMBL1745778 0.83 NNMT (0.52) NNMTSMN1; SMN2L3MBTL1KDM4EF7
SCHEMBL669121 0.83 NNMT (0.52) NNMTSMN1; SMN2L3MBTL1KDM4EF7
SCHEMBL23193160 0.81 NNMT (0.50) NNMTSMN1; SMN2L3MBTL1KDM4EF7
SCHEMBL1968189 0.81 NNMT (0.50) NNMTSMN1; SMN2L3MBTL1KDM4EF7
SCHEMBL17294856 0.79 NNMT (0.44) NNMTSMN1; SMN2L3MBTL1KDM4E
SCHEMBL1244783 0.79 SMN1; SMN2 (0.56) NNMTSMN1; SMN2L3MBTL1KDM4ETSHR
SCHEMBL30033603 0.79 AR (0.49) NNMTSMN1; SMN2L3MBTL1KDM4EF7
SCHEMBL4499172 0.76 NNMT (0.46) NNMTSMN1; SMN2L3MBTL1F7F3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257539-A1 SUBSTITUTED 4-HYDROXYPYRIMIDINE-5-CARBOXAMIDES Merck Sharp & Dohme Corp. (US) 2010-12-08 EP disclosed
WO-2009117269-A1 SUBSTITUTED 4-HYDROXYPYRIMIDINE-5-CARBOXAMIDES MERCK & CO., INC. (US) 2009-09-24 WO disclosed